The role of nitric oxide in the PKA inhibitor induced spatial memory deficits in rat: involvement of choline acetyltransferase

Eur J Pharmacol. 2013 Aug 15;714(1-3):478-85. doi: 10.1016/j.ejphar.2013.06.039. Epub 2013 Jul 5.

Abstract

Several lines of evidence show that cAMP-PKA signaling pathway plays critical role in memory functions and suggest nitric oxide as an important modulator in learning and memory. In this study, we assessed the effects of intra-hippocampal infusion of H-89, a selective PKAII inhibitor, and 1400 W, a selective inducible nitric oxide synthase (iNOS) inhibitor, on spatial memory in rats. By using the Morris water maze, spatial memory retention parameters were examined 48 h after the infusions through measuring escape latency, traveled distance, and swimming speed. The rats receiving intra-hippocampal infusions of 1400 W (100 µM/side) showed a significant reduction (*P<0.05) in escape latency and traveled distance in comparison with the control saline group. In contrast, a significant increase (**P<0.01) in escape latency and traveled distance was observed after infusion of 10 µM H-89. Moreover, among combination groups, co-administration of 1400 W (400 µM/side) with 10 µM/side of H-89 caused a significant reduction (*P<0.05) in escape latency and traveled distance in comparison with the H-89 group. Also, we evaluated the molecular effects of 1400 W on the expression of choline acetyltransferase (ChAT), a cholinergic marker, in the CA1 region of the hippocampus and medial septal area (MSA). Immunohistochemical analysis of post-training bilateral intra-hippocampal infusion of 1400 W revealed a significant increase in ChAT immunoreactivity levels in both the CA1 and the MSA regions. Overall, the results suggest that 1400 W has protective effect against H89-induced spatial memory impairment. Moreover, the observed memory improvements caused by 1400 W infusions, might be due to interaction of iNOS with the cholinergic system.

Keywords: Inducible nitric oxide synthase; Morris water maze; Protein kinase A; Spatial memory.

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • Animals
  • Choline O-Acetyltransferase / metabolism*
  • Cyclic AMP Response Element-Binding Protein / metabolism
  • Cyclic AMP-Dependent Protein Kinases / antagonists & inhibitors*
  • Drug Interactions
  • Escape Reaction / drug effects
  • Escape Reaction / physiology
  • Gene Expression Regulation, Enzymologic / drug effects
  • Hippocampus / drug effects
  • Hippocampus / metabolism
  • Hippocampus / physiology
  • Imines / pharmacology
  • Isoquinolines / pharmacology
  • Male
  • Maze Learning / drug effects
  • Maze Learning / physiology
  • Memory / drug effects*
  • Nitric Oxide / metabolism*
  • Phosphorylation / drug effects
  • Protein Kinase Inhibitors / pharmacology*
  • Rats
  • Rats, Wistar
  • Septal Nuclei / drug effects
  • Septal Nuclei / metabolism
  • Septal Nuclei / physiology
  • Spatial Behavior / drug effects*
  • Spatial Behavior / physiology*
  • Sulfonamides / pharmacology
  • Swimming

Substances

  • Cyclic AMP Response Element-Binding Protein
  • Imines
  • Isoquinolines
  • N-((3-(aminomethyl)phenyl)methyl)ethanimidamide
  • Protein Kinase Inhibitors
  • Sulfonamides
  • Nitric Oxide
  • Choline O-Acetyltransferase
  • Cyclic AMP-Dependent Protein Kinases
  • N-(2-(4-bromocinnamylamino)ethyl)-5-isoquinolinesulfonamide