β(3R3)-Peptides: design and synthesis of novel peptidomimetics and their self-assembling properties at the air-water interface

Org Biomol Chem. 2013 Sep 7;11(33):5399-403. doi: 10.1039/c3ob41135d.

Abstract

In this study we present the design and synthesis of a novel class of peptidomimetics, the β(3R3)-peptides. Via alternating directions of the amide bonds along β-peptide sequences, β(3R3)-peptides can potentially extend the structural space available to β-peptidic foldamers. Detailed analysis at the air-water interface shows strand conformations and the formation of sheet assemblies with different degrees of crystallinity. Furthermore β(3R3)-peptides exhibit a high proteolytic stability thus making them an interesting new class of peptidomimetics for biomedical applications.

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • Air
  • Molecular Conformation
  • Peptides / chemical synthesis*
  • Peptides / chemistry
  • Peptidomimetics / chemical synthesis*
  • Peptidomimetics / chemistry
  • Protein Structure, Secondary
  • Water / chemistry*

Substances

  • Peptides
  • Peptidomimetics
  • Water