Regulation of lipid and glucose homeostasis by mango tree leaf extract is mediated by AMPK and PI3K/AKT signaling pathways

Food Chem. 2013 Dec 1;141(3):2896-905. doi: 10.1016/j.foodchem.2013.05.121. Epub 2013 Jun 4.

Abstract

Ethanolic extract of Mangifera indica (mango) dose-dependently decreased serum glucose and triglyceride in KK-A(y) mice. Our in vitro and in vivo investigations revealed that the effect of mango leave extract (ME) on glucose and lipid homeostasis is mediated, at least in part, through the PI3K/AKT and AMPK signaling pathway. ME up-regulated the expression of PI3K, AKT and GYS genes by 2.0-fold, 3.2-fold, and 2.7-fold, respectively, leading to a decrease in glucose level. On the other hand, ME up-regulated AMPK and altered lipid metabolism. ME also down-regulated ACC (2.8-fold), HSL (1.6-fold), FAS (1.8-fold) and PPAR-γ (4.0-fold). Finally, we determined that active metabolites of benzophenone C-glucosides, Iriflophenone 3-C-β-glucoside and Foliamangiferoside A from ME, may play a dominant role in this integrated regulation of sugar and lipid homeostasis.

Keywords: 3T3-L1 cells; AMPK signaling pathway; Glucose and lipid regulation; Mangifera indica; PI3K/AKT signaling pathway.

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • 3T3-L1 Cells
  • AMP-Activated Protein Kinases / genetics
  • AMP-Activated Protein Kinases / metabolism
  • Animals
  • Female
  • Glucose / metabolism*
  • Glucose Metabolism Disorders / drug therapy*
  • Glucose Metabolism Disorders / enzymology
  • Glucose Metabolism Disorders / genetics
  • Glucose Metabolism Disorders / metabolism*
  • Homeostasis / drug effects*
  • Humans
  • Lipid Metabolism / drug effects*
  • Male
  • Mangifera / chemistry*
  • Mice
  • Mice, Inbred C57BL
  • Oncogene Protein v-akt / genetics
  • Oncogene Protein v-akt / metabolism
  • PPAR gamma / genetics
  • PPAR gamma / metabolism
  • Phosphatidylinositol 3-Kinases / genetics
  • Phosphatidylinositol 3-Kinases / metabolism
  • Plant Extracts / administration & dosage*
  • Plant Extracts / chemistry
  • Plant Leaves / chemistry
  • Signal Transduction / drug effects*
  • Trees / chemistry
  • Triglycerides / metabolism

Substances

  • PPAR gamma
  • Plant Extracts
  • Triglycerides
  • Phosphatidylinositol 3-Kinases
  • Oncogene Protein v-akt
  • AMP-Activated Protein Kinases
  • Glucose