A novel peptide inhibitor attenuates C-reactive protein's pro-inflammatory effects in-vivo

Int J Cardiol. 2013 Oct 9;168(4):3909-12. doi: 10.1016/j.ijcard.2013.06.047. Epub 2013 Jul 19.

Abstract

Background: Higher levels of C-reactive protein (CRP) predict cardiovascular events and also portend a poorer prognosis in patients with acute coronary syndromes. Much in-vitro and in-vivo data support a role for CRP in atherogenesis.

Methods: Using the one-bead-one-compound (OBOC) combinatorial library method we have successfully identified peptides against human CRP that inhibit its biological effects in-vitro. Hence we tested the effect of the best characterized inhibitor (CRP-i2) on the effects of CRP in an appropriate animal model, Wistar rats.

Results: Treatment with CRP resulted in significant increase in superoxide anion, nuclear factor kappaB (NFκb) activity and the release of biomarkers of inflammation from macrophages compared to Wistar rats treated with human albumin (HuSA). Pre-treatment with the inhibitor, CRP-i2, resulted in a significant reduction in CRP induced superoxide anion, NFκb activity and biomarkers of inflammation. Also, there were no observed clinical or laboratory related adverse effects.

Conclusions: We demonstrate that our novel peptide inhibitor attenuates the proinflammatory effects of CRP in-vivo. Future studies will examine the long-term effects of this inhibitor on vascular pathobiology.

Keywords: CRP; Inflammation; Macrophages.

Publication types

  • Research Support, N.I.H., Extramural

MeSH terms

  • Animals
  • C-Reactive Protein / antagonists & inhibitors*
  • C-Reactive Protein / metabolism*
  • C-Reactive Protein / toxicity
  • Humans
  • Inflammation / blood*
  • Inflammation / prevention & control
  • Inflammation Mediators / antagonists & inhibitors*
  • Inflammation Mediators / blood*
  • Peptide Fragments / pharmacology*
  • Peptide Fragments / therapeutic use
  • Rats
  • Rats, Wistar

Substances

  • Inflammation Mediators
  • Peptide Fragments
  • C-Reactive Protein