Polyhydrated ionogen with MgBr2 accelerates in vitro respiratory epithelial healing

Am J Rhinol Allergy. 2013 Jul-Aug;27(4):333-7. doi: 10.2500/ajra.2013.25.3910.

Abstract

Background: Remucoslization of the sinonasal cavity after sinus surgery is critical for successful outcomes. Recently, a novel antiprotease and antifibroblast compound, polyhydrated ionogen (PHI) with MgBr2, showed improved wound healing in a rabbit maxillary sinus mucosal wound model. We set out to determine if this effect was reproducible in an in vitro respiratory epithelial culture system.

Methods: Fully differentiated mature murine nasal septal air-liquid interface cultures were injured by creating a full-thickness 400-mM-wide scratch through the monolayer. Cultures were then treated with nothing, saline, or PHI with MgBr2 for 1 hour on the apical surface. Twenty-four hours after the injury cultures were fixed and processed for immunofluorescence with type IV beta-tubulin and Hoechst stain.

Results: Initial injury resulted in a wound of 394 micromolar (377-411 micromoler; 95% CI; n = 8). After 24 hours with no intervention the wound closed to 161 micromolar (138-184 micromolar; 95% CI; n = 9) and treatment with saline resulted in a residual gap of 88 micromolar (60-116 micromolar; 95% CI; n = 9; p < 0.05) and treatment with PHI with MgBr2 resulted in a gap of only 30 micromolar (14-46 micromolar; 95% CI; n = 9; p < 0.05).

Conclusion: Poor healing of the sinonasal mucosa after surgery with loss of ciliary function results in adverse clinical outcomes. In an in vitro sinonasal respiratory epithelial injury model, a one-time treatment with PHI with MgBr2 showed significantly improved wound healing compared with saline or nothing. This is a viable model to further investigate the mechanism by which PHI with MgBr2 improves sinonasal remucosolization.

Publication types

  • Comparative Study

MeSH terms

  • Animals
  • Bromides / pharmacology*
  • Cell Culture Techniques
  • Chronic Disease
  • Citrates / pharmacology
  • Disease Models, Animal
  • Magnesium / pharmacology*
  • Mice
  • Nasal Mucosa / drug effects*
  • Protease Inhibitors / administration & dosage
  • Rabbits
  • Respiratory Mucosa / drug effects
  • Rhinitis / surgery
  • Rubidium / pharmacology*
  • Sinusitis / surgery
  • Sodium Chloride / pharmacology*
  • Wound Healing / drug effects
  • Zinc / pharmacology*

Substances

  • Bromides
  • Citrates
  • PHI-5 formulation
  • Protease Inhibitors
  • Sodium Chloride
  • Magnesium
  • Zinc
  • Rubidium