Leflunomide plus oral prednisone in treatment of idiopathic membranous nephropathy: a retrospective clinical study of efficacy and safety

Nephrology (Carlton). 2013 Sep;18(9):615-22. doi: 10.1111/nep.12143.

Abstract

Aim: Treatment of idiopathic membranous nephropathy (IMN) remains a controversial issue. While clinical trials have shown that some immunosuppressants combined with glucocorticoid have a good efficacy on IMN patients. However, there is little data on leflunomide (LEF) in treatment of IMN.

Methods: Records of every patient with biopsy-proven IMN in Department of Nephrology, the First Affiliated Hospital, Xi'an Jiaotong University from January 2005 to December 2011 (n=194) were retrospectively analyzed. Patients with nephrotic IMN were treated with LEF plus oral prednisone (n=32) for at least 12 months, whereas 31 patients who did not receive any immunosuppressants were used as controls.

Results: Remission rates in the LEF group were 31.3%, 59.4%, 68.8% and 71.9% at 6, 9, 12 and 15 months, respectively, which were significantly higher than those in controls. In the LEF group, proteinuria decreased from 6.79 g/24 h at baseline to 5.63 g/24 h (P<0.01), 3.85 g/24 h (P<0.01) and 2.51 g/24 h (P<0.01) after treatment for 6, 9 and 12 months, respectively. Relapse occurred in five (21.7%) patients within a median of 14 months (range, 8-27) after cessation of LEF. No patients developed renal insufficiency during the therapeutic period. Multivariate analysis suggested that age negatively correlated with achievement of remission (odds ratio, 0.87; P<0.05). No serious adverse events were observed.

Conclusion: LEF plus oral prednisone may be an alternative treatment option in Chinese patients with nephrotic IMN.

Keywords: leflunomide; membranous nephropathy; nephrotic syndrome; prednisone; proteinuria.

MeSH terms

  • Administration, Oral
  • Adolescent
  • Adult
  • Aged
  • Biopsy
  • China
  • Drug Therapy, Combination
  • Female
  • Glomerulonephritis, Membranous / complications
  • Glomerulonephritis, Membranous / diagnosis
  • Glomerulonephritis, Membranous / drug therapy*
  • Glucocorticoids / administration & dosage*
  • Glucocorticoids / adverse effects
  • Hospitals, University
  • Humans
  • Immunosuppressive Agents / administration & dosage*
  • Immunosuppressive Agents / adverse effects
  • Isoxazoles / administration & dosage*
  • Isoxazoles / adverse effects
  • Leflunomide
  • Logistic Models
  • Male
  • Middle Aged
  • Multivariate Analysis
  • Odds Ratio
  • Prednisone / administration & dosage*
  • Prednisone / adverse effects
  • Proteinuria / drug therapy
  • Proteinuria / etiology
  • Recurrence
  • Remission Induction
  • Retrospective Studies
  • Risk Factors
  • Time Factors
  • Treatment Outcome
  • Young Adult

Substances

  • Glucocorticoids
  • Immunosuppressive Agents
  • Isoxazoles
  • Leflunomide
  • Prednisone