Epsilon aminocaproic acid prevents bleeding in severely thrombocytopenic patients with hematological malignancies

Cancer. 2013 Nov 1;119(21):3784-7. doi: 10.1002/cncr.28253. Epub 2013 Aug 6.

Abstract

Background: Despite prophylactic platelet transfusions, bleeding remains a significant problem in thrombocytopenic patients.

Methods: The antifibrinolytic agent epsilon aminocaproic acid (EACA) was administered to 44 chronically (median duration, 273 days) and severely (platelet count, 8 × 10(9)/L; range, 1 × 10(9)/L-19 × 10(9)/L) thrombocytopenic patients with hematological malignancies. Prophylactic EACA at a dose of 1 g twice daily was orally administered for a median duration of 47 days (range, 7 days-209 days) until the platelet count recovered to > 30; × 10(9) /L. Platelets were only transfused if bleeding occurred.

Results: While receiving EACA, 59% of the patients did not bleed, 25% had 19 episodes of spontaneously resolving minor bleeding that did not require platelet transfusion, and 16% received a median of 4 platelet transfusions (range, 1 transfusion-8 transfusions) for 1 major traumatic and 9 spontaneous grade 2 to grade 3 bleeding (based on the World Health Organization classification of idiopathic thrombocytopenic purpura). No EACA toxicities were noted, and venous thromboses were not observed.

Conclusions: EACA is well tolerated and is associated with a low risk of major bleeding in patients with hematological malignancies who are experiencing chronic severe thrombocytopenia.

Keywords: antifibrinolytic agent; bleeding; epsilon aminocaproic acid; hematologic malignancies; thrombocytopenia.

MeSH terms

  • Administration, Oral
  • Adolescent
  • Adult
  • Aged
  • Aged, 80 and over
  • Aminocaproic Acid / administration & dosage
  • Aminocaproic Acid / therapeutic use*
  • Antifibrinolytic Agents / administration & dosage
  • Antifibrinolytic Agents / therapeutic use*
  • Clinical Trials as Topic / statistics & numerical data
  • Drug Administration Schedule
  • Female
  • Hematologic Neoplasms / complications
  • Hematologic Neoplasms / drug therapy*
  • Hematologic Neoplasms / epidemiology
  • Hemorrhage / epidemiology
  • Hemorrhage / etiology
  • Hemorrhage / prevention & control*
  • Hemorrhage / therapy
  • Humans
  • Male
  • Middle Aged
  • Platelet Transfusion / statistics & numerical data
  • Retrospective Studies
  • Severity of Illness Index
  • Thrombocytopenia / complications
  • Thrombocytopenia / drug therapy*
  • Thrombocytopenia / epidemiology
  • Young Adult

Substances

  • Antifibrinolytic Agents
  • Aminocaproic Acid