Synthesis of peptides using tert-butyloxycarbonyl (Boc) as the α-amino protection group

Methods Mol Biol. 2013:1047:65-80. doi: 10.1007/978-1-62703-544-6_4.

Abstract

The use of the tert-butyloxycarbonyl (Boc) as the Nα-amino protecting group in peptide synthesis can be advantageous in several cases, such as synthesis of hydrophobic peptides and peptides containing ester and thioester moieties. The primary challenge of using Boc SPPS is the need for treatment of the resin-bound peptide with hazardous hydrogen fluoride (HF), which requires special equipment.

MeSH terms

  • Amino Acids / chemistry*
  • Formic Acid Esters / chemistry*
  • Peptides / chemical synthesis*
  • Solid-Phase Synthesis Techniques / methods

Substances

  • Amino Acids
  • Formic Acid Esters
  • Peptides
  • t-butyloxycarbonyl group