New pharmacokinetic methods. III. Two simple test for "deep pool effect"

J Clin Pharmacol. 1990 Aug;30(8):680-5. doi: 10.1002/j.1552-4604.1990.tb03626.x.

Abstract

If a portion of administered drug is distributed into a "deep" peripheral compartment, the drug's actual elimination half-life during the terminal exponential phase of elimination may be longer than determined by a single dose study or a tracer dose study ("deep pool effect"). Two simple methods of testing for "deep pool effect" applicable to drugs with either linear or nonlinear pharmacokinetic properties are described. The methods are illustrated with stable isotope labeled (13C15N2) tracer dose studies of phenytoin. No significant (P less than .05) "deep pool" effect was detected.

Publication types

  • Research Support, U.S. Gov't, Non-P.H.S.
  • Research Support, U.S. Gov't, P.H.S.

MeSH terms

  • Carbon Radioisotopes
  • Humans
  • Metabolic Clearance Rate
  • Pharmacokinetics*
  • Time Factors

Substances

  • Carbon Radioisotopes