Investigations into the mechanism by which sodium fluoride stimulates prostaglandin production in guinea-pig uterus

J Reprod Fertil. 1990 Jul;89(2):753-9. doi: 10.1530/jrf.0.0890753.

Abstract

Sodium fluoride (10 mM) caused a slow increase in the outputs of PGF-2 alpha, 6-keto-PGF-1 alpha and, to a lesser extent, PGE-2 from the Day-7 and Day-15 guinea-pig uterus superfused in vitro. This stimulatory action of sodium fluoride was not prevented by using calcium-free Krebs' solution. There was also a faster stimulation of 6-keto-PGF-1 alpha output from the Day-7 guinea-pig uterus produced by sodium fluoride, and this quicker response was abolished by using calcium-free Krebs' solution. TMB-8 (an intracellular calcium antagonist) inhibited the stimulatory action of sodium fluoride on the outputs of PGF-2 alpha, PGE-2 and 6-keto-PGF-1 alpha from the Day-7 guinea-pig uterus. W-7 and trifluoperazine (calmodulin antagonists) and neomycin (an inhibitor of phospholipase C) had no inhibitory effect on the increases in outputs of PGF-2 alpha, PGE-2 and 6-keto-PGF-1 alpha from the Day-7 guinea-pig uterus produced by sodium fluoride. These results indicate that sodium fluoride slowly stimulates uterine PGF-2 alpha, PGE-2 and 6-keto-PGF-1 alpha synthesis in the guinea-pig uterus by mobilizing intracellular calcium by a mechanism which apparently does not involve the activation of phospholipase C or the participation of calmodulin (or a related compound). The initial, faster stimulation of 6-keto-PGF-1 alpha synthesis in the Day-7 guinea-pig uterus by sodium fluoride is dependent upon extracellular calcium.

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • 6-Ketoprostaglandin F1 alpha / biosynthesis
  • Animals
  • Calcium Channel Blockers / pharmacology
  • Dinoprost / biosynthesis
  • Dinoprostone / biosynthesis
  • Female
  • Gallic Acid / analogs & derivatives
  • Gallic Acid / pharmacology
  • Guinea Pigs
  • Neomycin / pharmacology
  • Organ Culture Techniques
  • Prostaglandins / biosynthesis*
  • Sodium Fluoride / pharmacology*
  • Stimulation, Chemical
  • Trifluoperazine / pharmacology
  • Uterus / drug effects
  • Uterus / metabolism*

Substances

  • Calcium Channel Blockers
  • Prostaglandins
  • Trifluoperazine
  • 8-(N,N-diethylamino)octyl-3,4,5-trimethoxybenzoate
  • 6-Ketoprostaglandin F1 alpha
  • Gallic Acid
  • Sodium Fluoride
  • Dinoprost
  • Neomycin
  • Dinoprostone