Conformational transition of membrane-associated terminally acylated HIV-1 Nef

Structure. 2013 Oct 8;21(10):1822-33. doi: 10.1016/j.str.2013.08.008. Epub 2013 Sep 12.

Abstract

Many proteins are posttranslationally modified by acylation targeting them to lipid membranes. While methods such as X-ray crystallography and nuclear magnetic resonance are available to determine the structure of folded proteins in solution, the precise position of folded domains relative to a membrane remains largely unknown. We used neutron and X-ray reflection methods to measure the displacement of the core domain of HIV Nef from lipid membranes upon insertion of the N-terminal myristate group. Nef is one of several HIV-1 accessory proteins and an essential factor in AIDS progression. Upon insertion of the myristate and residues from the N-terminal arm, Nef transitions from a closed-to-open conformation that positions the core domain 70 Å from the lipid headgroups. This work rules out previous speculation that the Nef core remains closely associated with the membrane to optimize interactions with the cytoplasmic domain of MHC-1.

Publication types

  • Research Support, N.I.H., Extramural
  • Research Support, Non-U.S. Gov't
  • Research Support, U.S. Gov't, Non-P.H.S.

MeSH terms

  • Acylation
  • Adsorption
  • Amino Acid Motifs
  • HIV-1*
  • Membranes, Artificial
  • Models, Molecular
  • Neutron Diffraction
  • Phosphatidylglycerols / chemistry
  • Protein Processing, Post-Translational
  • Protein Structure, Tertiary
  • X-Ray Diffraction
  • nef Gene Products, Human Immunodeficiency Virus / chemistry*

Substances

  • Membranes, Artificial
  • Phosphatidylglycerols
  • nef Gene Products, Human Immunodeficiency Virus
  • nef protein, Human immunodeficiency virus 1
  • 1,2-dipalmitoylphosphatidylglycerol