[Effects of imatinib mesylate on the levels of endocrine hormones]

Zhonghua Xue Ye Xue Za Zhi. 2013 Sep;34(9):762-6. doi: 10.3760/cma.j.issn.0253-2727.2013.09.006.
[Article in Chinese]

Abstract

Objective: To measure the levels of hormones in chronic myelogenous leukemia (CML) patients receiving imatinib mesylate (IM) and evaluate the effects of IM on endocrine system.

Methods: 69 patients with CML while taking IM were enrolled and a total of 86 peripheral blood samples were detected. The levels of total triiodothyronine (TT3), total tetraiodothyronine (TT4), thyroid stimulating hormone (TSH), testosterone, progesterone, estradiol (E2), plasma total cortisol (PTC) at 8:00-10:00 am measured. Concentration of hormones in different groups were measured to evaluate the effects of IM on endocrine system and relationships with its administration duration, plasma concentration and clinical symptoms.

Results: (1) Of the 7 types of hormones, an elevation of TSH level was found in 14 patients (20.3%), a decrease of TT3 and testosterone in 8 patients (11.6%) and 8 males (18.6%), respectively. (2) A significant decline of TT3 and testosterone was observed in all patients divided by different administration duration. Negative correlation was seen between TT3 level and duration of administration (r=-0.273, P=0.010), which was also found for testosterone (r=-0.302, P=0.025). (3) There was no correlation between serum levels of the seven hormones and concentration of IM.

Conclusion: IM affect the levels of thyroid and sex hormones in some patients with clinical manifestations: a decrease of TT3, testosterone and testosterone, an increase of TSH, which have relationship with the duration of administration.

Publication types

  • English Abstract

MeSH terms

  • Adolescent
  • Adult
  • Aged
  • Aged, 80 and over
  • Benzamides / administration & dosage*
  • Benzamides / blood
  • Benzamides / therapeutic use
  • Female
  • Humans
  • Imatinib Mesylate
  • Leukemia, Myelogenous, Chronic, BCR-ABL Positive / blood*
  • Leukemia, Myelogenous, Chronic, BCR-ABL Positive / drug therapy
  • Male
  • Middle Aged
  • Piperazines / administration & dosage*
  • Piperazines / blood
  • Piperazines / therapeutic use
  • Pyrimidines / administration & dosage*
  • Pyrimidines / blood
  • Pyrimidines / therapeutic use
  • Thyrotropin / blood*
  • Triiodothyronine / blood*
  • Young Adult

Substances

  • Benzamides
  • Piperazines
  • Pyrimidines
  • Triiodothyronine
  • Imatinib Mesylate
  • Thyrotropin