Effects of N-acetylcysteine in ozone-induced chronic obstructive pulmonary disease model

PLoS One. 2013 Nov 18;8(11):e80782. doi: 10.1371/journal.pone.0080782. eCollection 2013.

Abstract

Introduction: Chronic exposure to high levels of ozone induces emphysema and chronic inflammation in mice. We determined the recovery from ozone-induced injury and whether an antioxidant, N-acetylcysteine (NAC), could prevent or reverse the lung damage.

Methods: Mice were exposed to ozone (2.5 ppm, 3 hours/12 exposures, over 6 weeks) and studied 24 hours (24h) or 6 weeks (6W) later. Nac (100 mg/kg, intraperitoneally) was administered either before each exposure (preventive) or after completion of exposure (therapeutic) for 6 weeks.

Results: After ozone exposure, there was an increase in functional residual capacity, total lung volume, and lung compliance, and a reduction in the ratio of forced expiratory volume at 25 and 50 milliseconds to forced vital capacity (FEV25/FVC, FEV50/FVC). Mean linear intercept (Lm) and airway hyperresponsiveness (AHR) to acetylcholine increased, and remained unchanged at 6W after cessation of exposure. Preventive NAC reduced the number of BAL macrophages and airway smooth muscle (ASM) mass. Therapeutic NAC reversed AHR, and reduced ASM mass and apoptotic cells.

Conclusion: Emphysema and lung function changes were irreversible up to 6W after cessation of ozone exposure, and were not reversed by NAC. The beneficial effects of therapeutic NAC may be restricted to the ASM.

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • 8-Hydroxy-2'-Deoxyguanosine
  • Acetylcysteine / administration & dosage
  • Acetylcysteine / pharmacology*
  • Animals
  • Apoptosis
  • Bronchial Hyperreactivity / chemically induced
  • Bronchoalveolar Lavage Fluid / chemistry
  • Bronchoalveolar Lavage Fluid / cytology
  • Deoxyguanosine / analogs & derivatives
  • Deoxyguanosine / blood
  • Disease Models, Animal
  • Emphysema / pathology
  • Expectorants / administration & dosage
  • Expectorants / pharmacology*
  • Gene Expression
  • Lung / drug effects
  • Lung / metabolism
  • Lung / pathology
  • Lung / physiopathology
  • Malondialdehyde / metabolism
  • Mice
  • Ozone / adverse effects*
  • Pulmonary Disease, Chronic Obstructive / chemically induced*
  • Pulmonary Disease, Chronic Obstructive / pathology
  • Pulmonary Disease, Chronic Obstructive / prevention & control*
  • Respiratory Function Tests

Substances

  • Expectorants
  • Malondialdehyde
  • Ozone
  • 8-Hydroxy-2'-Deoxyguanosine
  • Deoxyguanosine
  • Acetylcysteine