Ultrasound-promoted one-pot, four-component synthesis of pyridin-2(1H)-one derivatives

Molecules. 2013 Nov 25;18(12):14519-28. doi: 10.3390/molecules181214519.

Abstract

An efficient one-pot synthesis of 1,6-diamino-2-oxo-1,2,3,4-tetrahydro- pyridine-3,5-dicarbonitrile derivatives by four-component piperidine-catalyzed reactions of a ketone, malononitrile, ethyl cyanoacetate and hydrazine hydrate under ultrasound irradiation is described. This method provides several advantages such as shorter reaction times, excellent yields, and a simple workup procedure.

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • Molecular Structure
  • Nuclear Magnetic Resonance, Biomolecular
  • Pyridines / chemical synthesis
  • Pyridines / chemistry*
  • Sound*

Substances

  • Pyridines
  • pyridine