Properties of 5- and/or 2-modified 2'-O-cyanoethyl uridine residue: 2'-O-cyanoethyl-5-propynyl-2-thiouridine as an efficient duplex stabilizing component

Org Biomol Chem. 2014 Feb 21;12(7):1157-62. doi: 10.1039/c3ob41983e.

Abstract

We systematically synthesized eight types of 5- and/or 2-modified uridine derivatives and evaluated their effect on duplex stability. The incorporation of 2'-O-cyanoethyl-2-thio-5-propynyluridine (p(5)s(2)UOCE) into RNA was significantly effective for stabilization of RNA/RNA (+8.5 °C) and DNA/RNA (+10.4 °C) duplexes. These striking effects were maintained in oligonucleotides with different sequences or multiple incorporations. In addition, p(5)s(2)UOCE increased selectivity toward the correct AU Watson-Crick base pair over the most stable mismatched base pair in both RNA/RNA and DNA/RNA duplexes. Hence, p(5)s(2)UOCE could be useful for various applications of modified oligonucleotides that need high duplex stability and base pairing selectivity.

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • DNA / chemistry*
  • Nucleic Acid Conformation
  • RNA / chemistry*
  • Thiouridine / analogs & derivatives*
  • Thiouridine / chemistry
  • Uridine / analogs & derivatives
  • Uridine / chemical synthesis*
  • Uridine / chemistry

Substances

  • Thiouridine
  • RNA
  • DNA
  • Uridine