Both glimepiride and high-dose metformin are important for sustained glucose lowering in Japanese type 2 diabetes patients on glimepiride-sitagliptin-metformin therapy: subanalysis of a single-center, open-label, randomized study

Diabetes Technol Ther. 2014 Jul;16(7):442-6. doi: 10.1089/dia.2013.0310. Epub 2014 Feb 14.

Abstract

Background: In a previous single-center, open-label randomized 3-month study of triple oral antidiabetes drug (OAD) therapy, we investigated factors affecting the glycemic control afforded by sitagliptin, high-dose metformin, and low-dose glimepiride. Patients were prospectively assigned to either Group 1 (50% reduction in metformin) or Group 2 (discontinuation of glimepiride) and compared. The results showed that the glycated hemoglobin (HbA1c) levels of patients in Group 2 deteriorated more than those in Group 1, whereas HbA1c levels were maintained in some patients in both groups.

Materials and methods: To determine the factors associated with maintenance of HbA1c under this triple OAD regimen, data from the prospective study were further analyzed.

Results: In both Groups 1 and 2, the baseline HbA1c level was higher in patients with HbA1c ≥7.0% after 3 months of treatment than those with an HbA1c level of <7.0%. A generalized linear model revealed that high-dose metformin was associated with a deterioration of HbA1c levels in Group 2.

Conclusions: Together, the findings indicate that glimepiride and high-dose metformin are important for sustained glycemic control in triple OAD therapy with sitagliptin, metformin, and sulfonylurea.

Publication types

  • Randomized Controlled Trial

MeSH terms

  • Administration, Oral
  • Aged
  • Aged, 80 and over
  • Asian People / statistics & numerical data
  • Blood Glucose / drug effects*
  • Blood Glucose / metabolism
  • Diabetes Mellitus, Type 2 / blood
  • Diabetes Mellitus, Type 2 / drug therapy*
  • Drug Therapy, Combination
  • Female
  • Glycated Hemoglobin / drug effects*
  • Glycated Hemoglobin / metabolism
  • Humans
  • Hypoglycemic Agents / therapeutic use*
  • Japan
  • Male
  • Metformin / therapeutic use*
  • Middle Aged
  • Prospective Studies
  • Pyrazines / therapeutic use*
  • Sitagliptin Phosphate
  • Sulfonylurea Compounds / therapeutic use*
  • Treatment Outcome
  • Triazoles / therapeutic use*

Substances

  • Blood Glucose
  • Glycated Hemoglobin A
  • Hypoglycemic Agents
  • Pyrazines
  • Sulfonylurea Compounds
  • Triazoles
  • hemoglobin A1c protein, human
  • glimepiride
  • Metformin
  • Sitagliptin Phosphate