Cinnamon extract improves insulin sensitivity in the brain and lowers liver fat in mouse models of obesity

PLoS One. 2014 Mar 18;9(3):e92358. doi: 10.1371/journal.pone.0092358. eCollection 2014.

Abstract

Objectives: Treatment of diabetic subjects with cinnamon demonstrated an improvement in blood glucose concentrations and insulin sensitivity but the underlying mechanisms remained unclear. This work intends to elucidate the impact of cinnamon effects on the brain by using isolated astrocytes, and an obese and diabetic mouse model.

Methods: Cinnamon components (eugenol, cinnamaldehyde) were added to astrocytes and liver cells to measure insulin signaling and glycogen synthesis. Ob/ob mice were supplemented with extract from cinnamomum zeylanicum for 6 weeks and cortical brain activity, locomotion and energy expenditure were evaluated. Insulin action was determined in brain and liver tissues.

Results: Treatment of primary astrocytes with eugenol promoted glycogen synthesis, whereas the effect of cinnamaldehyde was attenuated. In terms of brain function in vivo, cinnamon extract improved insulin sensitivity and brain activity in ob/ob mice, and the insulin-stimulated locomotor activity was improved. In addition, fasting blood glucose levels and glucose tolerance were greatly improved in ob/ob mice due to cinnamon extracts, while insulin secretion was unaltered. This corresponded with lower triglyceride and increased liver glycogen content and improved insulin action in liver tissues. In vitro, Fao cells exposed to cinnamon exhibited no change in insulin action.

Conclusions: Together, cinnamon extract improved insulin action in the brain as well as brain activity and locomotion. This specific effect may represent an important central feature of cinnamon in improving insulin action in the brain, and mediates metabolic alterations in the periphery to decrease liver fat and improve glucose homeostasis.

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • Acrolein / analogs & derivatives*
  • Acrolein / pharmacology
  • Acrolein / therapeutic use
  • Adiposity / drug effects
  • Animals
  • Astrocytes / drug effects
  • Brain / drug effects*
  • Brain / metabolism
  • Cell Line
  • Cinnamomum zeylanicum / chemistry
  • Energy Intake
  • Eugenol / pharmacology*
  • Eugenol / therapeutic use
  • Glycogen / biosynthesis
  • Humans
  • Insulin / administration & dosage
  • Insulin / physiology
  • Insulin Resistance
  • Liver / drug effects*
  • Liver / metabolism
  • Male
  • Mice
  • Mice, Inbred C57BL
  • Mice, Obese
  • Motor Activity / drug effects
  • Obesity / drug therapy
  • Obesity / metabolism*
  • Plant Extracts / pharmacology*
  • Plant Extracts / therapeutic use

Substances

  • Insulin
  • Plant Extracts
  • Eugenol
  • Acrolein
  • Glycogen
  • cinnamaldehyde

Grants and funding

The project was supported in part by grants from the German Federal Ministry of Education and Research (BMBF) to the German Center for Diabetes Research (DZD e.V.; 01GI0925). Additional parts of the funding are internal department funds of the University of Tuebingen (employment of people at the University of Tuebingen). The funders had no role in study design, data collection and analysis, decision to publish, or preparation of the manuscript.