Abstract
Tumor endothelial cells (ECs) promote cancer progression in ways beyond their role as conduits supporting metabolism. However, it is unknown how vascular niche-derived paracrine factors, defined as angiocrine factors, provoke tumor aggressiveness. Here, we show that FGF4 produced by B cell lymphoma cells (LCs) through activating FGFR1 upregulates the Notch ligand Jagged1 (Jag1) on neighboring ECs. In turn, upregulation of Jag1 on ECs reciprocally induces Notch2-Hey1 in LCs. This crosstalk enforces aggressive CD44(+)IGF1R(+)CSF1R(+) LC phenotypes, including extranodal invasion and chemoresistance. Inducible EC-selective deletion of Fgfr1 or Jag1 in the Eμ-Myc lymphoma model or impairing Notch2 signaling in mouse and human LCs diminished lymphoma aggressiveness and prolonged mouse survival. Thus, targeting the angiocrine FGF4-FGFR1/Jag1-Notch2 loop inhibits LC aggressiveness and enhances chemosensitivity.
Copyright © 2014 Elsevier Inc. All rights reserved.
Publication types
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Research Support, N.I.H., Extramural
MeSH terms
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Animals
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Burkitt Lymphoma / genetics
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Burkitt Lymphoma / metabolism*
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Burkitt Lymphoma / pathology*
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Calcium-Binding Proteins / genetics
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Calcium-Binding Proteins / metabolism*
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Cell Cycle Proteins / metabolism
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Cell Proliferation
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Drug Resistance, Neoplasm*
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Endothelial Cells / metabolism
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Enzyme Activation
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Fibroblast Growth Factor 4 / metabolism*
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Genes, myc
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Humans
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Hyaluronan Receptors / metabolism
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Intercellular Signaling Peptides and Proteins / genetics
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Intercellular Signaling Peptides and Proteins / metabolism*
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Jagged-1 Protein
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Membrane Proteins / genetics
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Membrane Proteins / metabolism*
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Mice
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Mice, Transgenic
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Neoplasm Invasiveness
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RNA Interference
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RNA, Small Interfering
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Receptor, Fibroblast Growth Factor, Type 1 / metabolism*
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Receptor, IGF Type 1 / metabolism
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Receptor, Macrophage Colony-Stimulating Factor / metabolism
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Receptor, Notch2 / metabolism*
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Serrate-Jagged Proteins
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Signal Transduction / genetics
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Tumor Cells, Cultured
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Up-Regulation
Substances
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Calcium-Binding Proteins
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Cell Cycle Proteins
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Fibroblast Growth Factor 4
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Hey1 protein, mouse
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Hyaluronan Receptors
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Intercellular Signaling Peptides and Proteins
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JAG1 protein, human
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Jag1 protein, mouse
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Jagged-1 Protein
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Membrane Proteins
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RNA, Small Interfering
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Receptor, Notch2
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Serrate-Jagged Proteins
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Receptor, Fibroblast Growth Factor, Type 1
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Receptor, IGF Type 1
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Receptor, Macrophage Colony-Stimulating Factor