Synthesis of RNA oligomer using 9-fluorenylmethoxycarbonyl (Fmoc) group for 5'-hydroxyl protection

Nucleic Acids Symp Ser. 1988:(19):13-6.

Abstract

An approach using a new combination of protecting groups in RNA oligomer synthesis is proposed, in which 5'-hydroxyl group of ribose moiety is temporarily protected with the alkaline labile 9-fluorenylmethoxycarbonyl (Fmoc) group and the 2'-hydroxyl group is protected with the acid labile 1-ethoxyethyl (EE) group. The adoption of this method presented great selectivity in removing the 5'-hydroxyl protecting group and facilitated the RNA oligomer synthesis. A RNA pentamer was synthesized by the phosphotriester method in solution.

MeSH terms

  • Chromatography, High Pressure Liquid
  • Fluorenes
  • Hydroxylation
  • Indicators and Reagents
  • Oligoribonucleotides / chemical synthesis*
  • Oligoribonucleotides / isolation & purification
  • RNA / chemical synthesis*

Substances

  • Fluorenes
  • Indicators and Reagents
  • Oligoribonucleotides
  • RNA