A pilot study comparing the effect of flaxseed, aromatase inhibitor, and the combination on breast tumor biomarkers

Nutr Cancer. 2014;66(4):566-75. doi: 10.1080/01635581.2014.894097. Epub 2014 Mar 26.

Abstract

Use of complementary approaches is common among breast cancer survivors. Potential interactions between aromatase inhibitors (AI) and high phytoestrogen foods, such as flaxseed (FS), are not often described. We conducted a pilot 2 × 2 factorial, randomized intervention study between tumor biopsy and resection, in 24 postmenopausal women with estrogen receptor positive (ER+) breast cancer, to assess the effects of FS and anastrozole, and possible interactions between them, on serum steroid hormone and tumor-related characteristics associated with long-term survival (Roswell Park Cancer Institute, 2007-2010). The effect of each treatment vs. placebo on outcomes was determined by linear regression adjusting for pretreatment measure, stage, and grade. Although not statistically significant, mean ERβ expression was approximately 40% lower from pre- to postintervention in the FS + AI group only. We observed a statistically significant negative association (β ± SE -0.3 ± 0.1; P = 0.03) for androstenedione in the FS + AI group vs. placebo and for DHEA with AI treatment (β ± SE -1.6 ± 0.6; P = 0.009). Enterolactone excretion was much lower in the FS + AI group compared to the FS group. Our results do not support strong effects of FS on AI activity for selected breast tumor characteristics or serum steroid hormone levels but suggest AI therapy might reduce the production of circulating mammalian lignans from FS.

Trial registration: ClinicalTrials.gov NCT00612560.

Publication types

  • Randomized Controlled Trial
  • Research Support, N.I.H., Extramural

MeSH terms

  • Adolescent
  • Adult
  • Aged
  • Aged, 80 and over
  • Anastrozole
  • Aromatase Inhibitors / pharmacology*
  • Biomarkers, Tumor / blood*
  • Body Mass Index
  • Breast Neoplasms / blood
  • Breast Neoplasms / drug therapy*
  • Estrogen Receptor beta / genetics
  • Estrogen Receptor beta / metabolism
  • Female
  • Flax / chemistry*
  • Gonadal Steroid Hormones / blood
  • Humans
  • Lignans / urine
  • Linear Models
  • Middle Aged
  • Nitriles / pharmacology
  • Pilot Projects
  • Treatment Outcome
  • Triazoles / pharmacology
  • Young Adult

Substances

  • Aromatase Inhibitors
  • Biomarkers, Tumor
  • Estrogen Receptor beta
  • Gonadal Steroid Hormones
  • Lignans
  • Nitriles
  • Triazoles
  • Anastrozole

Associated data

  • ClinicalTrials.gov/NCT00612560