Redox-triggered C-C coupling of diols and alkynes: synthesis of β,γ-unsaturated α-hydroxyketones and furans by ruthenium-catalyzed hydrohydroxyalkylation

Angew Chem Int Ed Engl. 2014 Mar 17;53(12):3232-5. doi: 10.1002/anie.201311130.

Abstract

Direct ruthenium-catalyzed CC coupling of alkynes and vicinal diols to form β,γ-unsaturated ketones occurs with complete levels of regioselectivity and good to complete control over the alkene geometry. Exposure of the reaction products to substoichiometric quantities of p-toluenesulfonic acid induces cyclodehydration to form tetrasubstituted furans. These alkyne-diol hydrohydroxyalkylations contribute to a growing body of merged redox-construction events that bypass the use of premetalated reagents and, hence, stoichiometric quantities of metallic by-products.

Publication types

  • Research Support, N.I.H., Extramural
  • Research Support, Non-U.S. Gov't

MeSH terms

  • Alkynes / chemistry*
  • Catalysis
  • Cyclization
  • Furans / chemical synthesis*
  • Ketones / chemical synthesis*
  • Molecular Structure
  • Oxidation-Reduction
  • Ruthenium / chemistry*
  • Stereoisomerism

Substances

  • Alkynes
  • Furans
  • Ketones
  • Ruthenium