Antibody ligation of CM1 on cisplatin-exposed HeLa cells induces apoptosis through reactive oxygen species-dependent Fas ligand expression

Int J Oncol. 2014 Jun;44(6):2016-24. doi: 10.3892/ijo.2014.2361. Epub 2014 Mar 27.

Abstract

Centrocyte/centroblast marker 1 (CM1) has been identified as a pro-apoptosis molecule on B-cell lymphoma cells as well as several types of cancer cells. In this study, we investigated its signaling mechanism in HeLa cells after treatment with cisplatin in order to potentially identify a new therapeutic target. The CM1 molecule was induced on the surface of cisplatin-exposed HeLa cells. In these cells, ligation of CM1 with anti-CM1 monoclonal antibodies inhibited cell proliferation and produced reactive oxygen species. Fas ligand (FasL) expression was upregulated without upregulating Fas in cisplatin-exposed HeLa cells after CM1 stimulation. Pretreatment with N-acetylcysteine, a pan-capase inhibitor, and ZB4, an antagonistic anti-Fas antibody, effectively inhibited the apoptotic effect triggered by CM1. CM1 ligation induced apoptosis through disruption of the mitochondrial membrane potential, decreased Bcl-2 and phosphorylated ERK expression. These findings identify CM1 as a potential new therapeutic target related to cisplatin-exposed cervical cancer.

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • Acetylcysteine / pharmacology
  • Antibodies, Monoclonal / metabolism*
  • Antibodies, Monoclonal / pharmacology
  • Apoptosis / genetics
  • Apoptosis / physiology
  • Apoptosis Regulatory Proteins / metabolism*
  • Cell Proliferation / genetics
  • Cisplatin / pharmacology*
  • Fas Ligand Protein / metabolism*
  • Gene Expression Regulation, Neoplastic
  • HeLa Cells / drug effects*
  • Humans
  • Membrane Potential, Mitochondrial / drug effects
  • Membrane Potential, Mitochondrial / genetics
  • Membrane Potential, Mitochondrial / physiology
  • Reactive Oxygen Species / metabolism*
  • fas Receptor / antagonists & inhibitors
  • fas Receptor / metabolism

Substances

  • Antibodies, Monoclonal
  • Apoptosis Regulatory Proteins
  • FAS protein, human
  • Fas Ligand Protein
  • Reactive Oxygen Species
  • centrocyte centroblast marker 1 protein, human
  • fas Receptor
  • Cisplatin
  • Acetylcysteine