Dynamic contrast-enhanced MRI parameters as biomarkers for the effect of vatalanib in patients with non-small-cell lung cancer

Future Oncol. 2014 Apr;10(5):823-33. doi: 10.2217/fon.13.248.

Abstract

Aims: To assess the utility of dynamic contrast-enhanced MRI parameters in the demonstration of early antiangiogenic effects and as prognostic biomarkers in second-line treatment of advanced-stage non-small-cell lung cancer with vatalanib.

Patients & methods: The transfer constant (K(trans)) and the initial area under the contrast concentration-time curve at 60 s (AUC60) were assessed in 46 patients. Changes were compared with response evaluation from computed tomography imaging and Response Evaluation Criteria In Solid Tumors guidelines.

Results: Statistically significant mean reductions in K(trans) (38.4%; p < 0.0001) and AUC60 (24.9%; p < 0.0001) were found at day 2. After 12 weeks, 16 patients (35%) demonstrated stable disease and 30 (65%) demonstrated progressive disease. No statistically significant differences in day 2 K(trans) and AUC60 reductions between stable disease and progressive disease patients were found.

Conclusion: Dynamic contrast-enhanced MRI can demonstrate a statistically significant reduction in vascular parameters of non-small-cell lung cancer, but does not predict patient outcome.

MeSH terms

  • Aged
  • Angiogenesis Inhibitors / administration & dosage*
  • Biomarkers*
  • Carcinoma, Non-Small-Cell Lung / diagnostic imaging
  • Carcinoma, Non-Small-Cell Lung / drug therapy*
  • Carcinoma, Non-Small-Cell Lung / pathology
  • Clinical Trials as Topic
  • Contrast Media / administration & dosage
  • Contrast Media / therapeutic use
  • Drug Evaluation
  • Drug-Related Side Effects and Adverse Reactions / pathology
  • Female
  • Humans
  • Magnetic Resonance Imaging*
  • Male
  • Middle Aged
  • Neoplasm Staging
  • Phthalazines / administration & dosage*
  • Phthalazines / adverse effects
  • Pyridines / administration & dosage*
  • Pyridines / adverse effects
  • Radiography

Substances

  • Angiogenesis Inhibitors
  • Biomarkers
  • Contrast Media
  • Phthalazines
  • Pyridines
  • vatalanib