DDI-CPI, a server that predicts drug-drug interactions through implementing the chemical-protein interactome

Nucleic Acids Res. 2014 Jul;42(Web Server issue):W46-52. doi: 10.1093/nar/gku433. Epub 2014 May 29.

Abstract

Drug-drug interactions (DDIs) may cause serious side-effects that draw great attention from both academia and industry. Since some DDIs are mediated by unexpected drug-human protein interactions, it is reasonable to analyze the chemical-protein interactome (CPI) profiles of the drugs to predict their DDIs. Here we introduce the DDI-CPI server, which can make real-time DDI predictions based only on molecular structure. When the user submits a molecule, the server will dock user's molecule across 611 human proteins, generating a CPI profile that can be used as a feature vector for the pre-constructed prediction model. It can suggest potential DDIs between the user's molecule and our library of 2515 drug molecules. In cross-validation and independent validation, the server achieved an AUC greater than 0.85. Additionally, by investigating the CPI profiles of predicted DDI, users can explore the PK/PD proteins that might be involved in a particular DDI. A 3D visualization of the drug-protein interaction will be provided as well. The DDI-CPI is freely accessible at http://cpi.bio-x.cn/ddi/.

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • Drug Design*
  • Humans
  • Internet
  • Molecular Docking Simulation
  • Pharmaceutical Preparations / chemistry
  • Proteins / chemistry*
  • Proteins / drug effects
  • Sertraline / chemistry
  • Software*

Substances

  • Pharmaceutical Preparations
  • Proteins
  • Sertraline