Proposal of an in silico profiler for categorisation of repeat dose toxicity data of hair dyes

Arch Toxicol. 2015 May;89(5):733-41. doi: 10.1007/s00204-014-1277-8. Epub 2014 Jun 3.

Abstract

This study outlines the analysis of 94 chemicals with repeat dose toxicity data taken from Scientific Committee on Consumer Safety opinions for commonly used hair dyes in the European Union. Structural similarity was applied to group these chemicals into categories. Subsequent mechanistic analysis suggested that toxicity to mitochondria is potentially a key driver of repeat dose toxicity for chemicals within each of the categories. The mechanistic hypothesis allowed for an in silico profiler consisting of four mechanism-based structural alerts to be proposed. These structural alerts related to a number of important chemical classes such as quinones, anthraquinones, substituted nitrobenzenes and aromatic azos. This in silico profiler is intended for grouping chemicals into mechanism-based categories within the adverse outcome pathway paradigm.

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • Computer Simulation*
  • Data Interpretation, Statistical
  • Hair Dyes / chemistry
  • Hair Dyes / toxicity*
  • Humans
  • Mitochondria / drug effects
  • Models, Biological
  • Structure-Activity Relationship

Substances

  • Hair Dyes