Rescue therapy with adefovir in decompensated liver cirrhosis patients with lamivudine-resistant hepatitis B virus

Clin Mol Hepatol. 2014 Jun;20(2):168-76. doi: 10.3350/cmh.2014.20.2.168. Epub 2014 Jun 30.

Abstract

Background/aims: Adefovir dipivoxil (ADV) is a nucleotide analogue that is effective against lamivudine-resistant hepatitis B virus (HBV). The aim of this study was to determine the long-term clinical outcomes after ADV rescue therapy in decompensated patients infected with lamivudine-resistant HBV.

Methods: In total, 128 patients with a decompensated state and lamivudine-resistant HBV were treated with ADV at a dosage of 10 mg/day for a median of 33 months in this multicenter cohort study.

Results: Following ADV treatment, 86 (72.3%) of 119 patients experienced a decrease in Child-Pugh score of at least 2 points, and the overall end-stage liver disease score decreased from 16±5 to 14±10 (mean ± SD, P<0.001) during the follow-up period. With ADV treatment, 67 patients (56.3%) had undetectable serum HBV DNA (detection limit, 0.5 pg/mL). Virologic breakthrough occurred in 38 patients (36.1%) and 9 patients had a suboptimal ADV response. The overall survival rate was 89.9% (107/119), and a suboptimal response to ADV treatment was associated with both no improvement in Child-Pugh score (≥2 points; P=0.001) and high mortality following ADV rescue therapy (P=0.012).

Conclusions: Three years of ADV treatment was effective and safe in decompensated patients with lamivudine-resistant HBV.

Keywords: Adefovir dipivoxil; Decompensation; Hepatitis B virus; Lamivudine-resistant.

Publication types

  • Multicenter Study
  • Research Support, Non-U.S. Gov't

MeSH terms

  • Adenine / analogs & derivatives*
  • Adenine / therapeutic use
  • Adult
  • Aged
  • Antiviral Agents / therapeutic use*
  • Cohort Studies
  • DNA, Viral / blood
  • Drug Resistance, Viral
  • Female
  • Hepatitis B / complications
  • Hepatitis B / drug therapy*
  • Hepatitis B e Antigens / blood
  • Hepatitis B virus / genetics
  • Humans
  • Lamivudine / therapeutic use*
  • Liver Cirrhosis / diagnosis*
  • Liver Cirrhosis / etiology
  • Liver Cirrhosis / mortality
  • Male
  • Middle Aged
  • Odds Ratio
  • Organophosphonates / therapeutic use*
  • Retrospective Studies
  • Severity of Illness Index
  • Survival Rate

Substances

  • Antiviral Agents
  • DNA, Viral
  • Hepatitis B e Antigens
  • Organophosphonates
  • Lamivudine
  • adefovir
  • Adenine