Studies on pharmacological activation of human serum immunoglobulin G by chemical modification and active subfragments. VIII. Effect of carboxamide-methylated light chain (Fr.I-L) on leukocyte functions

J Pharmacobiodyn. 1989 Mar;12(3):159-63. doi: 10.1248/bpb1978.12.159.

Abstract

Human serum immunoglobulin G light chain (Fr.I-L), which was reduced and carboxamide-methylated, showed no effect on formyl-methionyl-leucyl-phenylalanine (FMLP)-induced chemotaxis nor on phagocytosis of yeasts when directly added to guinea pig polymorphonuclear leukocytes (PMNs). However, intravenously administered Fr.I-L inhibited emigration of leukocytes into the peritoneal cavity and promoted phagocytosis of yeasts in a yeast-induced peritonitis model in mice. Moreover, Fr.I-L reduced FMLP-induced chemiluminescence (CL) from PMNs. These facts indicated that the anti-inflammatory action of Fr.I-L was caused by inhibiting emigration of leukocytes into the injured site and scavenging superoxide radicals from the cells.

MeSH terms

  • Animals
  • Chemical Phenomena
  • Chemistry
  • Chemotaxis, Leukocyte
  • Edema / immunology
  • Guinea Pigs
  • Humans
  • Immunoglobulin G / immunology*
  • Immunoglobulin Light Chains / immunology*
  • Iodoacetamide*
  • Iodoacetates*
  • Leukocytes / immunology*
  • Luminescent Measurements
  • Male
  • Methylation
  • Mice
  • Mice, Inbred ICR
  • Mycoses / immunology
  • N-Formylmethionine Leucyl-Phenylalanine / pharmacology
  • Neutrophils / immunology
  • Peritonitis / etiology
  • Peritonitis / immunology
  • Phagocytosis
  • Structure-Activity Relationship

Substances

  • Immunoglobulin G
  • Immunoglobulin Light Chains
  • Iodoacetates
  • N-Formylmethionine Leucyl-Phenylalanine
  • Iodoacetamide