Successful treatment of multiple intracranial meningiomas with the antiprogesterone receptor agent mifepristone (RU486)

Acta Neurochir (Wien). 2014 Oct;156(10):1831-5. doi: 10.1007/s00701-014-2188-4. Epub 2014 Jul 31.

Abstract

Background: Meningiomas are the most frequent primary brain tumor in adults. Evidence suggests that female sex hormones play a role in the meningioma tumorigenesis. In particular, progesterone, has a receptor (PR) that is highly expressed in the majority of grade I meningiomas. Multiple meningiomas (diffuse meningiomatosis) are less frequent, but have a higher female predominance and a higher PR expression. They are, therefore, attractive candidates for anti-PR therapy.

Methods: We treated three consecutive women with multiple meningiomas with mifepristone (RU 486). It is a synthetic steroid with high affinity for both progesterone and glucocorticoid receptors.

Results: The treatment was well tolerated, and we observed an important and long-lasting clinical (3/3) and radiological response (2/3) or stabilisation. All the three patients are now stable after five to nine years of treatment.

Conclusions: These encouraging results strongly support a prospective clinical trial in this preselected population.

Publication types

  • Case Reports
  • Research Support, Non-U.S. Gov't

MeSH terms

  • Female
  • Hormone Antagonists / administration & dosage
  • Hormone Antagonists / adverse effects
  • Hormone Antagonists / pharmacology*
  • Humans
  • Meningeal Neoplasms / drug therapy*
  • Meningeal Neoplasms / pathology
  • Meningeal Neoplasms / physiopathology
  • Meningioma / drug therapy*
  • Meningioma / pathology
  • Meningioma / physiopathology
  • Middle Aged
  • Mifepristone / administration & dosage
  • Mifepristone / adverse effects
  • Mifepristone / pharmacology*
  • Receptors, Progesterone / antagonists & inhibitors*
  • Treatment Outcome

Substances

  • Hormone Antagonists
  • Receptors, Progesterone
  • Mifepristone