[Effect of a calcium inhibitor, nicardipine, on aldosterone secretion in primary hyperaldosteronism]

Arch Mal Coeur Vaiss. 1989 Jul;82(7):1237-40.
[Article in French]

Abstract

The purpose of the study was to evaluate the effects of a dihydropyridine calcium antagonist, nicardipine (N), on blood pressure (BP) and aldosterone secretion in hypertensive patients (pt) with primary aldosteronism. The study concerned 8 pts, mean age 55.6 +/- 7.7 years, 1 pt with aldosterone-producing adenoma (APA) and 7 pts with idiopathic aldosteronism: plasma renin activity (PRA) and plasma aldosterone concentration (PAC) were respectively 0.30 +/- 0.2 ng/ml/h) and 314 +/- 109 pg/ml. Acute administration of 12 mg of nicardipine during 90 mn (three periods of N infusion during 30 mn: 0.4 mg/mn-5 mn; then 0.08 mg/mn-25 mn) significantly decreased BP, with an increase in heart rate (HR); the levels of PAC were significantly reduced with a slight but not significant increase in PRA, 60 mn after N: (table; see text) N decreased also PAC in the pt with APA [600 to 410 pg/ml] but did not improve hypokalemia (3.1 vs 3.3 mmol/l, n = 8 N.S.). In contrast, PAC levels were not modified 2 hours after acute oral administration of captopril (1 mg/kg): 302 +/- 164 pg/ml vs 332 +/- 191 pg/ml (NS). This study demonstrated the antihypertensive efficacy of acute infusion of nicardipine in primary aldosteronism; the decrease of PAC under this calcium antagonist suggested its potential interest in the management of idiopathic aldosteronism.

Publication types

  • Clinical Trial

MeSH terms

  • Aged
  • Aldosterone / metabolism*
  • Blood Pressure / drug effects
  • Clinical Trials as Topic
  • Drug Evaluation
  • Female
  • Humans
  • Hyperaldosteronism / metabolism*
  • Hypertension / drug therapy
  • Male
  • Middle Aged
  • Nicardipine / pharmacology*
  • Nicardipine / therapeutic use

Substances

  • Aldosterone
  • Nicardipine