Preparation and characterization of galactosylated alginate-chitosan oligomer microcapsule for hepatocytes microencapsulation

Carbohydr Polym. 2014 Nov 4:112:502-11. doi: 10.1016/j.carbpol.2014.06.025. Epub 2014 Jun 19.

Abstract

Galactosylated alginate (GA)-chitosan oligomer microcapsule was prepared to provide a sufficient mechanical stability, a selective permeability and an appropriate three-dimensional (3D) microenvironment for hepatocytes microencapsulation. The microcapsule has a unique asymmetric membrane structure, with a dense layer located in the inner surface and gradually decreasing toward the outside surface. The stable microcapsule was obtained when GA lower than 50%, while the permeability was increased with increasing of GA. A balance between mechanical stability and permeability was achieved through modulating membrane porosity and thickness. The optimal microcapsule displays a selective permeability allowing efficient transport of human serum albumin while effectively blocking immunoglobulin G. Hepatocytes exhibited high and long term viability (>92%), proliferability, multicellular spheroid morphology, and enhancement of liver-specific functions in the microcapsule wherein galactose moieties present chemical cues to support cell-matrix interactions while the 3D structure of the microcapsule behaves physical cues to facilitate cell-cell interactions.

Keywords: Galactosylated alginate; Hepatocytes; Mechanical stability; Microcapsule; Microenvironment; Selective permeability.

Publication types

  • Research Support, N.I.H., Extramural
  • Research Support, Non-U.S. Gov't

MeSH terms

  • Alginates / chemistry*
  • Capsules / chemistry
  • Cell Proliferation
  • Cell Survival
  • Cells, Cultured
  • Chemistry Techniques, Synthetic
  • Chitosan / chemistry*
  • Drug Carriers
  • Drug Compounding / methods*
  • Galactose / chemistry
  • Glucuronic Acid / chemistry
  • Hepatocytes / chemistry
  • Hepatocytes / cytology*
  • Hexuronic Acids / chemistry
  • Humans
  • Magnetic Resonance Spectroscopy
  • Permeability
  • Porosity
  • Serum Albumin / chemistry
  • Serum Albumin / metabolism
  • Serum Albumin / pharmacokinetics

Substances

  • Alginates
  • Capsules
  • Drug Carriers
  • Hexuronic Acids
  • Serum Albumin
  • Glucuronic Acid
  • Chitosan
  • Galactose