Phosphorylation of ribosomal protein S6 mediates compensatory renal hypertrophy

Kidney Int. 2015 Mar;87(3):543-56. doi: 10.1038/ki.2014.302. Epub 2014 Sep 17.

Abstract

The molecular mechanism underlying renal hypertrophy and progressive nephron damage remains poorly understood. Here we generated congenic ribosomal protein S6 (rpS6) knock-in mice expressing nonphosphorylatable rpS6 and found that uninephrectomy-induced renal hypertrophy was significantly blunted in these knock-in mice. Uninephrectomy-induced increases in cyclin D1 and decreases in cyclin E in the remaining kidney were attenuated in the knock-in mice compared with their wild-type littermates. Uninephrectomy induced rpS6 phosphorylation in the wild-type mice; however, no rpS6 phosphorylation was detected in uninephrectomized or sham-operated knock-in mice. Nonetheless, uninephrectomy stimulated comparable 4E-BP1 phosphorylation in both knock-in and wild-type mice, indicating that mTORC1 was still activated in the knock-in mice. Moreover, the mTORC1 inhibitor rapamycin prevented both rpS6 and 4E-BP1 phosphorylation, significantly blunted uninephrectomy-induced renal hypertrophy in wild-type mice, but did not prevent residual renal hypertrophy despite inhibiting 4E-BP1 phosphorylation in uninephrectomized knock-in mice. Thus, both genetic and pharmacological approaches unequivocally demonstrate that phosphorylated rpS6 is a downstream effector of the mTORC1-S6K1 signaling pathway mediating renal hypertrophy. Hence, rpS6 phosphorylation facilitates the increase in cyclin D1 and decrease in cyclin E1 that underlie the hypertrophic nature of uninephrectomy-induced kidney growth.

Publication types

  • Research Support, N.I.H., Extramural
  • Research Support, Non-U.S. Gov't

MeSH terms

  • Adaptor Proteins, Signal Transducing
  • Animals
  • Carrier Proteins / metabolism*
  • Cell Cycle Proteins
  • Cyclin D1 / metabolism
  • Cyclin E / metabolism
  • Cyclin-Dependent Kinase 2 / metabolism
  • Cyclin-Dependent Kinase 4 / metabolism
  • Eukaryotic Initiation Factors
  • Female
  • Gene Knock-In Techniques
  • Hypertrophy / etiology
  • Hypertrophy / metabolism
  • Kidney / metabolism*
  • Kidney / pathology*
  • Male
  • Mechanistic Target of Rapamycin Complex 1
  • Mice
  • Multiprotein Complexes / metabolism
  • Nephrectomy* / adverse effects
  • Oncogene Proteins / metabolism
  • Phosphoproteins / metabolism*
  • Phosphorylation / drug effects
  • Ribosomal Protein S6 / genetics
  • Ribosomal Protein S6 / metabolism*
  • Ribosomal Protein S6 Kinases, 90-kDa / metabolism
  • Signal Transduction / drug effects
  • Signal Transduction / genetics
  • Sirolimus / pharmacology
  • TOR Serine-Threonine Kinases / metabolism

Substances

  • Adaptor Proteins, Signal Transducing
  • Carrier Proteins
  • Ccnd1 protein, mouse
  • Cell Cycle Proteins
  • Cyclin E
  • Eif4ebp1 protein, mouse
  • Eukaryotic Initiation Factors
  • Multiprotein Complexes
  • Oncogene Proteins
  • Phosphoproteins
  • Ribosomal Protein S6
  • cyclin E1, mouse
  • Cyclin D1
  • Mechanistic Target of Rapamycin Complex 1
  • Ribosomal Protein S6 Kinases, 90-kDa
  • Rps6ka1 protein, mouse
  • TOR Serine-Threonine Kinases
  • Cyclin-Dependent Kinase 2
  • Cyclin-Dependent Kinase 4
  • Sirolimus