Enhancer of zeste homolog 2 is widely expressed in T-cell neoplasms, is associated with high proliferation rate and correlates with MYC and pSTAT3 expression in a subset of cases

Leuk Lymphoma. 2015 Jul;56(7):2087-91. doi: 10.3109/10428194.2014.968780. Epub 2014 Oct 30.

Abstract

Enhancer of zeste homolog 2 (EZH2), an epigenetic regulator and H3k27-specific histone methyltransferase, is important for transcriptional regulation. EZH2 has been found to be overexpressed in B-cell lymphomas, as well as some T-cell lymphomas. Here we investigated the expression of EZH2 by immunohistochemical staining in a wide range of T-cell neoplasms. We found that EZH2 is highly expressed in all categories of T-cell neoplasia studied, and its expression strongly correlates with a high proliferation rate. Although up-regulation of EZH2 has been reported to be modulated by the pSTAT3-MYC pathway, our data indicate that EZH2 expression is correlated with MYC and/or pSTAT3 expression in only a subset of T-cell lymphomas, and that other mechanisms may control the overexpression of EZH2 in many T-cell lymphomas. The high level of EZH2 expression in T cell lymphomas suggest that these neoplasms may benefit from targeted treatment with a small molecule inhibitor of EZH2 currently in use in clinical trials.

Keywords: EZH2; MYC; T-cell lymphoma; pSTAT3; proliferation.

MeSH terms

  • Biomarkers, Tumor / metabolism*
  • Cell Proliferation*
  • Enhancer of Zeste Homolog 2 Protein
  • Humans
  • Immunoenzyme Techniques
  • Leukemia, T-Cell / metabolism
  • Leukemia, T-Cell / pathology*
  • Lymphoma, T-Cell / metabolism
  • Lymphoma, T-Cell / pathology*
  • Neoplasm Staging
  • Phosphorylation
  • Polycomb Repressive Complex 2 / metabolism*
  • Prognosis
  • Proto-Oncogene Proteins c-myc / metabolism*
  • STAT3 Transcription Factor / metabolism*
  • Up-Regulation

Substances

  • Biomarkers, Tumor
  • MYC protein, human
  • Proto-Oncogene Proteins c-myc
  • STAT3 Transcription Factor
  • STAT3 protein, human
  • EZH2 protein, human
  • Enhancer of Zeste Homolog 2 Protein
  • Polycomb Repressive Complex 2