Direct renin inhibitor therapy and swimming training: hemodynamic and cardiac effects in hypertensive and normotensive rats

Clin Exp Hypertens. 2015;37(4):345-52. doi: 10.3109/10641963.2014.972562. Epub 2014 Oct 27.

Abstract

Purpose: This study aimed to analyze the hemodynamic and cardiac effects of direct renin inhibitor (DRI) treatment and swimming training in hypertensive rats.

Methods: Seventy-seven rats were divide into eight groups: sedentary normotensive (SN), trained normotensive (TN), sedentary normotensive treated with DRI (SN_DRI), trained normotensive treated with DRI (TN_DRI), sedentary hypertensive (SH), trained hypertensive (TH), sedentary hypertensive treated with DRI (SH_DRI), trained hypertensive treated with DRI (TH_DRI). Swimming training occurred for up to 60 min, five times a week for four weeks. The hypertensive animals were treated with 20 mg ċ kg(-1) ċ day(-1) L-NAME for four weeks. Groups treated with DRI received 10 mg ċ kg(-1) ċ day(-1) of aliskiren for four weeks. After the treatment period, all the animals underwent femoral artery catheterization surgery for direct measurement of cardiovascular variables.

Results: The SH group presented hypertension (136.4 ± 5.0 mmHg) compared to the SN (107.1 ± 1.7 mmHg). The TH group showed lower mean arterial pressure (MAP) than the SH (121.1 ± 1.3 mmHg), but the treatment with DRI did not attenuate hypertension (128.2 ± 4.9 mmHg). The analysis of collagen areas demonstrated that treatment with DRI may attenuate cardiac remodeling in situations of hypertension, in the condition of treatment alone or combined with physical training.

Conclusion: Both interventions in combination may be more effective at reducing cardiovascular risk in hypertensive subjects.

Keywords: Arterial blood pressure; direct renin inhibitor; hypertension; physical training.

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • Amides / therapeutic use*
  • Animals
  • Blood Pressure / drug effects
  • Blood Pressure / physiology*
  • Disease Models, Animal
  • Enzyme Inhibitors / therapeutic use
  • Fumarates / therapeutic use*
  • Heart / physiopathology
  • Hypertension / blood
  • Hypertension / drug therapy*
  • Hypertension / physiopathology
  • Male
  • NG-Nitroarginine Methyl Ester / pharmacology*
  • Physical Conditioning, Animal / methods*
  • Rats
  • Rats, Wistar
  • Renin / antagonists & inhibitors*
  • Renin / blood
  • Risk Factors
  • Swimming / physiology*

Substances

  • Amides
  • Enzyme Inhibitors
  • Fumarates
  • aliskiren
  • Renin
  • NG-Nitroarginine Methyl Ester