Curcumin-induced histone acetylation inhibition improves stress-induced gastric ulcer disease in rats

Mol Med Rep. 2015 Mar;11(3):1911-6. doi: 10.3892/mmr.2014.2958. Epub 2014 Nov 14.

Abstract

Curcumin is known to possess anti‑inflammatory properties. Despite the fact that curcumin is known to be a strong inhibitor of H+, K+‑ATPase activity, the mechanism underlying the curcumin‑induced inhibition of the transcription of the H+, K+‑ATPase α subunit in gastric mucosal parietal cells remains unclear. The present study investigated the possible mechanism by which curcumin inhibits stomach H+, K+‑ATPase activity during the acute phase of gastric ulcer disease. A rat model of stress‑induced gastric ulcers was produced, in which the anti‑ulcer effects of curcumin were examined. Curcumin‑induced inhibition of the H+, K+‑ATPase promoter via histone acetylation, was verified using a chromatin immunoprecipitation assay. The results showed that curcumin improved stress‑induced gastric ulcer disease in rats, as demonstrated by increased pH values and reduced gastric mucosal hemorrhage and ulcer index. These effects were accompanied by a significant reduction in the level of histone H3 acetylation at the site of the H+, K+‑ATPase promoter and in the expression of the gastric H+,K+‑ATPase α subunit gene and protein. In conclusion, curcumin downregulated the acetylation of histone H3 at the site of the H+, K+‑ATPase promoter gene, thereby inhibiting the transcription and expression of the H+, K+‑ATPase gene. Curcumin was shown to have a preventive and therapeutic effect in gastric ulcer disease.

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • Acetylation / drug effects
  • Animals
  • Anti-Inflammatory Agents / administration & dosage
  • Anti-Inflammatory Agents / pharmacology*
  • Curcumin / administration & dosage
  • Curcumin / pharmacology*
  • Disease Models, Animal
  • Gastric Juice / chemistry
  • Gastric Juice / drug effects
  • Gastric Mucosa / drug effects
  • Gastric Mucosa / metabolism
  • Gastric Mucosa / pathology
  • Histones / metabolism*
  • Hydrogen-Ion Concentration / drug effects
  • Male
  • Promoter Regions, Genetic
  • RNA, Messenger / genetics
  • Rats
  • Sodium-Potassium-Exchanging ATPase / genetics
  • Sodium-Potassium-Exchanging ATPase / metabolism
  • Stomach Ulcer / drug therapy
  • Stomach Ulcer / etiology*
  • Stomach Ulcer / metabolism*
  • Stomach Ulcer / pathology
  • Stress, Physiological*
  • Stress, Psychological*

Substances

  • Anti-Inflammatory Agents
  • Histones
  • RNA, Messenger
  • Sodium-Potassium-Exchanging ATPase
  • Curcumin