Radical production in liver mitochondria by peroxidic tumor promoters

Biochem Biophys Res Commun. 1989 May 15;160(3):1067-72. doi: 10.1016/s0006-291x(89)80111-1.

Abstract

Eleven peroxides have been tested to determine if there is a correlation between tumor-promoting activity and the ability to stimulate radical production in mitochondria. When non-respiring rat liver mitochondria are treated with these peroxidic compounds in the presence of DMPO, ESR signals are observed from the spin trapping of carbon- and oxygen-centered radicals in the case of 4 of the 7 peroxides that are known to be tumor promoters. Enhancement of carbon-centered radical production is observed in the presence of respiratory substrate. Thus there does not appear to be a correlation between tumor-promoting activity of peroxidic compounds and radical production in mitochondria. Oxidants can act as promoters either by 1- or 2-electron oxidation pathways; both types of mechanisms may be inhibited by antioxidants, which can scavenge either radicals or electrophiles.

Publication types

  • Research Support, Non-U.S. Gov't
  • Research Support, U.S. Gov't, P.H.S.

MeSH terms

  • Animals
  • Carcinogens / pharmacology*
  • Cyclic N-Oxides / pharmacology
  • Electron Spin Resonance Spectroscopy
  • Electron Transport
  • Free Radicals
  • Male
  • Mitochondria, Liver / drug effects
  • Mitochondria, Liver / metabolism*
  • Oxidation-Reduction
  • Oxygen / metabolism
  • Peroxides / pharmacology*
  • Rats
  • Rats, Inbred Strains

Substances

  • Carcinogens
  • Cyclic N-Oxides
  • Free Radicals
  • Peroxides
  • 5,5-dimethyl-1-pyrroline-1-oxide
  • Oxygen