Alpha-chloralose opens the chloride channel of frog isolated sensory neurons

Brain Res. 1989 Sep 25;498(1):181-4. doi: 10.1016/0006-8993(89)90418-6.

Abstract

The effect of alpha-chloralose on the sensory neurons isolated enzymatically and mechanically from frog dorsal root ganglia was studied using a suction-pipette technique. The threshold concentration of alpha-chloralose was around 3 x 10(-5) M and the current produced by alpha-chloralose saturated at the concentration of 3 x 10(-3) M or more. The dose-response curve for alpha-chloralose provided a Ka value of 6 x 10(-4) M and a Hill coefficient of 1.8. The reversal potential of the response elicited by alpha-chloralose was close to the equilibrium potential for Cl- (ECl), indicating that the current was carried through Cl- channels. The current-voltage relationship indicated that there was little voltage dependence in the alpha-chloralose-induced response. The analysis of the variance of the alpha-chloralose-induced Cl- current fluctuations showed two types of the receptor-ionophore complexes with different channel conductances.

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • Animals
  • Chloralose / pharmacology*
  • Chloride Channels
  • Chlorides
  • Ganglia, Spinal / drug effects
  • Ganglia, Spinal / physiology*
  • In Vitro Techniques
  • Membrane Potentials / drug effects
  • Membrane Proteins / physiology*
  • Neurons, Afferent / drug effects
  • Neurons, Afferent / physiology*
  • Rana catesbeiana

Substances

  • Chloride Channels
  • Chlorides
  • Membrane Proteins
  • Chloralose