Vascular type I aldosterone binding sites are physiological mineralocorticoid receptors

Endocrinology. 1989 Oct;125(4):2224-6. doi: 10.1210/endo-125-4-2224.

Abstract

In vitro, Type I receptors have high and equivalent affinity for aldosterone, corticosterone and cortisol: in vivo, physiological mineralocorticoid target tissues (kidney, colon, parotid) are highly aldosterone-selective, in contrast with hippocampus and heart. In the present study we show that the mesenteric vascular arcade is similarly highly aldosterone-selective in vivo, and in vitro shows considerable levels of 11 beta OH steroid dehydrogenase activity, previously postulated as the mechanism whereby glucocorticoids are excluded from physiological mineralocorticoid receptors.

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • 11-beta-Hydroxysteroid Dehydrogenases
  • Aldosterone / metabolism*
  • Animals
  • Binding Sites
  • Blood Vessels / enzymology
  • Blood Vessels / metabolism
  • Hydroxysteroid Dehydrogenases / metabolism
  • Male
  • Mineralocorticoids / metabolism
  • Rats
  • Rats, Inbred Strains
  • Receptors, Mineralocorticoid
  • Receptors, Steroid / metabolism*
  • Splanchnic Circulation*

Substances

  • Mineralocorticoids
  • Receptors, Mineralocorticoid
  • Receptors, Steroid
  • Aldosterone
  • Hydroxysteroid Dehydrogenases
  • 11-beta-Hydroxysteroid Dehydrogenases