β-1 tubulin R307H SNP alters microtubule dynamics and affects severity of a hereditary thrombocytopenia

J Thromb Haemost. 2015 Apr;13(4):651-9. doi: 10.1111/jth.12824. Epub 2015 Jan 22.

Abstract

Background: Single nucleotide polymorphisms (SNPs) in platelet-associated genes partly explain inherent variability in platelet counts. Patients with monoallelic Bernard Soulier syndrome due to the Bolzano mutation (GPIBA A156V) have variable platelet counts despite a common mutation for unknown reasons.

Objectives: We investigated the effect of the most common SNP (R307H) in the hematopoietic-specific tubulin isotype β-1 in these Bernard Soulier patients and potential microtubule-based mechanisms of worsened thrombocytopenia.

Patients/methods: Ninety-four monoallelic Bolzano mutation patients were evaluated for the R307H β-1 SNP and had platelet counts measured by three methods; the Q43P SNP was also evaluated. To investigate possible mechanisms underlying this association, we used molecular modeling of β-1 tubulin with and without the R307H SNP. We transfected SNP or non-SNP β-1 tubulin into MCF-7 and CMK cell lines and measured microtubule regrowth after nocodazole-induced depolymerization.

Results: We found that patients with at least one R307H SNP allele had significantly worse thrombocytopenia; manual platelet counting revealed a median platelet count of 124 in non-SNP patients and 76 in SNP patients (both ×10(9) L(-1) ; P < 0.01). The Q43P SNP had no significant association with platelet count. Molecular modeling suggested a structural relationship between the R307H SNP and microtubule stability via alterations in the M-loop of β tubulin; in vitro microtubule recovery assays revealed that cells transfected with R307H SNP β-1 had significantly impaired microtubule recovery.

Conclusions: Our data show that the R307H SNP is significantly associated with the degree of thrombocytopenia in congenital and acquired platelet disorders, and may affect platelets by altering microtubule behavior.

Keywords: Bernard-Soulier syndrome; beta-tubulin; cytoskeleton; microtubules; polymorphism, single nucleotide.

Publication types

  • Research Support, N.I.H., Extramural
  • Research Support, Non-U.S. Gov't

MeSH terms

  • Bernard-Soulier Syndrome / blood
  • Bernard-Soulier Syndrome / diagnosis
  • Bernard-Soulier Syndrome / genetics*
  • Blood Platelets / drug effects
  • Blood Platelets / metabolism*
  • Crystallography, X-Ray
  • Genetic Markers
  • Genetic Predisposition to Disease
  • Humans
  • MCF-7 Cells
  • Microtubules / drug effects
  • Microtubules / metabolism*
  • Models, Molecular
  • Phenotype
  • Platelet Count
  • Polymorphism, Single Nucleotide*
  • Protein Conformation
  • Protein Stability
  • Severity of Illness Index
  • Structure-Activity Relationship
  • Transfection
  • Tubulin / chemistry
  • Tubulin / genetics*
  • Tubulin / metabolism*
  • Tubulin Modulators / pharmacology

Substances

  • Genetic Markers
  • TUBB1 protein, human
  • Tubulin
  • Tubulin Modulators