Synthesis of pyrazoles from 1,3-diols via hydrogen transfer catalysis

Org Lett. 2015 Mar 20;17(6):1405-8. doi: 10.1021/acs.orglett.5b00266. Epub 2015 Feb 26.

Abstract

1,3-Diols engage in ruthenium-catalyzed hydrogen transfer in the presence of alkyl hydrazines to provide 1,4-disubstituted pyrazoles. Regioselective synthesis of unsymmetrical pyrazoles from β-hydroxy ketones is also described.