Picodiscs for facile protein-glycolipid interaction analysis

Anal Chem. 2015 Apr 21;87(8):4402-8. doi: 10.1021/acs.analchem.5b00170. Epub 2015 Apr 9.

Abstract

Protein interactions with glycolipids are implicated in diverse cellular processes. However, the study of protein-glycolipid complexes remains a significant experimental challenge. Here, we describe a powerful new assay that combines electrospray ionization mass spectrometry (ESI-MS) and picodiscs, which are composed of human sphingolipid activator protein saposin A and a small number of phospholipids, to display glycolipids in a lipid environment for protein-glycolipid interaction studies in aqueous solution. Time-resolved measurements of enzyme catalyzed hydrolysis of glycolipid substrates and the detection of low, moderate, and high affinity protein-glycolipid interactions serve to demonstrate the reliability and versatility of the assay.

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • Glycolipids / chemistry*
  • Glycolipids / metabolism
  • Humans
  • Hydrolysis
  • Neuraminidase / chemistry
  • Neuraminidase / metabolism
  • Saposins / chemistry*
  • Saposins / metabolism
  • Spectrometry, Mass, Electrospray Ionization
  • Time Factors

Substances

  • Glycolipids
  • Saposins
  • Neu3 protein, human
  • Neuraminidase