Safety assessment of [3S, 3'S]-astaxanthin--Subchronic toxicity study in rats

Food Chem Toxicol. 2015 Jul:81:129-136. doi: 10.1016/j.fct.2015.04.017. Epub 2015 Apr 21.

Abstract

Astaxanthin, a naturally occurring xanthophyll, is commercially used as a coloring agent in salmon feed, but also marketed as a dietary supplement. The objective of this study was to investigate the subchronic toxicity of synthetic [3S, 3'S]-Astaxanthin in rats. A powder formulation containing approximately 20% [3S, 3'S]-Astaxanthin was administered via the diet to groups of 10 male and 10 female Wistar rats at concentrations of 5000, 15,000 and 50,000 ppm for a period of 13 weeks. A formulation of comparable composition but without [3S, 3'S]-Astaxanthin served as a placebo control. There were no effects observed on survival, clinical examinations, clinical pathology, estrous cycle as well as on sperm parameters. At terminal necropsy, a macroscopically visible brown-blue discoloration of the gastrointestinal contents was noted which was considered to be secondary to the violet-brown color of the test material. No other significant or dose-related abnormalities were found in the tissues collected at termination. Our observations support that ingestion of [3S, 3'S]-Astaxanthin of up to 700-920 mg/kg bw/day in rats in a gelatin/carbohydrate formulation is without adverse effects.

Keywords: Astaxanthin; Rat; Subchronic toxicity.

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • Alanine Transaminase / blood
  • Alkaline Phosphatase / blood
  • Animals
  • Aspartate Aminotransferases / blood
  • Bilirubin / blood
  • Blood Glucose / metabolism
  • Body Weight
  • Cholesterol / blood
  • Creatinine / blood
  • Dietary Supplements
  • Dose-Response Relationship, Drug
  • Drug Evaluation, Preclinical
  • Female
  • Male
  • Organ Size / drug effects
  • Rats
  • Rats, Wistar
  • Serum Albumin / metabolism
  • Toxicity Tests, Subchronic / methods*
  • Triglycerides / blood
  • Xanthophylls / blood
  • Xanthophylls / toxicity

Substances

  • Blood Glucose
  • Serum Albumin
  • Triglycerides
  • Xanthophylls
  • astaxanthine
  • Cholesterol
  • Creatinine
  • Aspartate Aminotransferases
  • Alanine Transaminase
  • Alkaline Phosphatase
  • Bilirubin