Central Fibroblast Growth Factor 21 Browns White Fat via Sympathetic Action in Male Mice

Endocrinology. 2015 Jul;156(7):2470-81. doi: 10.1210/en.2014-2001. Epub 2015 Apr 29.

Abstract

Fibroblast growth factor 21 (FGF21) has multiple metabolic actions, including the induction of browning in white adipose tissue. Although FGF21 stimulated browning results from a direct interaction between FGF21 and the adipocyte, browning is typically associated with activation of the sympathetic nervous system through cold exposure. We tested the hypothesis that FGF21 can act via the brain, to increase sympathetic activity and induce browning, independent of cell-autonomous actions. We administered FGF21 into the central nervous system via lateral ventricle infusion into male mice and found that the central treatment increased norepinephrine turnover in target tissues that include the inguinal white adipose tissue and brown adipose tissue. Central FGF21 stimulated browning as assessed by histology, expression of uncoupling protein 1, and the induction of gene expression associated with browning. These effects were markedly attenuated when mice were treated with a β-blocker. Additionally, neither centrally nor peripherally administered FGF21 initiated browning in mice lacking β-adrenoceptors, demonstrating that an intact adrenergic system is necessary for FGF21 action. These data indicate that FGF21 can signal in the brain to activate the sympathetic nervous system and induce adipose tissue thermogenesis.

Publication types

  • Research Support, N.I.H., Extramural

MeSH terms

  • Adipocytes, Brown / metabolism
  • Adipocytes, White / drug effects*
  • Adipocytes, White / metabolism
  • Adipose Tissue, Brown / metabolism*
  • Adipose Tissue, White / drug effects*
  • Adipose Tissue, White / metabolism
  • Adrenergic beta-Antagonists / pharmacology
  • Animals
  • Fibroblast Growth Factors / pharmacology*
  • Infusions, Intraventricular
  • Ion Channels / drug effects*
  • Ion Channels / metabolism
  • Male
  • Mice
  • Mice, Knockout
  • Mitochondrial Proteins / drug effects*
  • Mitochondrial Proteins / metabolism
  • Receptors, Adrenergic, beta / genetics*
  • Receptors, Adrenergic, beta-1 / genetics
  • Receptors, Adrenergic, beta-2 / genetics
  • Receptors, Adrenergic, beta-3 / genetics
  • Sympathetic Nervous System / drug effects*
  • Sympathetic Nervous System / metabolism
  • Thermogenesis
  • Uncoupling Protein 1

Substances

  • Adrenergic beta-Antagonists
  • Ion Channels
  • Mitochondrial Proteins
  • Receptors, Adrenergic, beta
  • Receptors, Adrenergic, beta-1
  • Receptors, Adrenergic, beta-2
  • Receptors, Adrenergic, beta-3
  • Ucp1 protein, mouse
  • Uncoupling Protein 1
  • fibroblast growth factor 21
  • Fibroblast Growth Factors