Extended-Release Niacin Versus Fenofibrate in HIV-Infected Participants With Low High-Density Lipoprotein Cholesterol: Effects on Endothelial Function, Lipoproteins, and Inflammation

Clin Infect Dis. 2015 Sep 1;61(5):840-9. doi: 10.1093/cid/civ385. Epub 2015 May 15.

Abstract

Background: Low levels of high-density lipoprotein cholesterol (HDL-C) are common in individuals with human immunodeficiency virus (HIV) infection, persist during antiretroviral therapy (ART), and are associated with increased cardiovascular disease (CVD) risk.

Methods: Virologically controlled participants without CVD on stable ART with low HDL-C (men <40 mg/dL, women <50 mg/dL) and triglycerides >150 mg/dL were randomized to receive open-label extended-release niacin 1500 mg/day with aspirin 325 mg/day or fenofibrate 200 mg/day for 24 weeks. The primary endpoint was the week 24 within-arm change in brachial artery flow-mediated dilation (FMD) in participants with complete follow-up scans.

Results: Of 99 participants, 74 had complete data (35 niacin, 39 fenofibrate). Median age was 45 years, 77% were male, median CD4(+) count was 561 cells/µL, and brachial FMD was 4.2%. Median HDL-C was 32 mg/dL for men and 38 mg/dL for women, low-density lipoprotein cholesterol was 103 mg/dL, and triglycerides were 232 mg/dL. In men, HDL-C increased a median of 3 mg/dL with niacin and 6.5 mg/dL with fenofibrate (P < .001 for both). In women, HDL-C increased a median of 16 mg/dL with niacin and 8 mg/dL with fenofibrate (P = .08 for both). After 24 weeks, there was no significant change in FMD in either arm; the median (interquartile range) change was +0.6% (-1.6 to 2.3) with niacin (P = .28) and +0.5% (-1.0 to 3.0) with fenofibrate (P = .19). Neither treatment significantly affected C-reactive protein, interleukin 6, or D-dimer levels.

Conclusions: Despite improvements in lipids, niacin or fenofibrate treatment for 24 weeks did not improve endothelial function or inflammatory markers in participants with well-controlled HIV infection and low HDL-C.

Clinical trials registration: NCT01426438.

Keywords: HIV; endothelial function; fenofibrate; high-density lipoprotein; niacin.

Publication types

  • Randomized Controlled Trial
  • Research Support, N.I.H., Extramural
  • Research Support, Non-U.S. Gov't

MeSH terms

  • Adult
  • Brachial Artery / physiology
  • C-Reactive Protein
  • Cholesterol, HDL / blood*
  • Delayed-Action Preparations
  • Dyslipidemias / complications
  • Dyslipidemias / drug therapy
  • Dyslipidemias / epidemiology
  • Endothelium, Vascular / drug effects
  • Female
  • Fenofibrate / administration & dosage
  • Fenofibrate / adverse effects
  • Fenofibrate / pharmacology*
  • Fenofibrate / therapeutic use*
  • HIV Infections / complications
  • HIV Infections / epidemiology*
  • Humans
  • Inflammation
  • Lipoproteins / blood
  • Male
  • Middle Aged
  • Niacin / administration & dosage
  • Niacin / adverse effects
  • Niacin / pharmacology*
  • Niacin / therapeutic use*

Substances

  • Cholesterol, HDL
  • Delayed-Action Preparations
  • Lipoproteins
  • Niacin
  • C-Reactive Protein
  • Fenofibrate

Associated data

  • ClinicalTrials.gov/NCT01426438