Localization of Hidden Insulinomas with ⁶⁸Ga-DOTA-Exendin-4 PET/CT: A Pilot Study

J Nucl Med. 2015 Jul;56(7):1075-8. doi: 10.2967/jnumed.115.157768. Epub 2015 May 21.

Abstract

(111)In-DOTA-exendin-4 SPECT/CT has been shown to be highly efficient in the detection of insulinomas. We aimed at determining whether novel PET/CT imaging with [Nle(14),Lys(40)(Ahx-DOTA-(68)Ga)NH2]exendin-4 ((68)Ga-DOTA-exendin-4) is feasible and sensitive in detecting benign insulinomas.

Methods: (68)Ga-DOTA-exendin-4 PET/CT and (111)In-DOTA-exendin-4 SPECT/CT were performed in a randomized cross-over order on 5 patients with endogenous hyperinsulinemic hypoglycemia. The gold standard for comparison was the histologic diagnosis after surgery.

Results: In 4 patients histologic diagnosis confirmed a benign insulinoma, whereas one patient refused surgery despite a positive (68)Ga-DOTA-exendin-4 PET/CT scan. In 4 of 5 patients, previously performed conventional imaging (CT or MR imaging) was not able to localize the insulinoma. (68)Ga-DOTA-exendin-4 PET/CT correctly identified the insulinoma in 4 of 4 patients, whereas (111)In-DOTA-exendin-4 SPECT/CT correctly identified the insulinoma in only 2 of 4 patients.

Conclusion: These preliminary data suggest that the use of (68)Ga-DOTA-exendin-4 PET/CT in detecting hidden insulinomas is feasible.

Keywords: 68Ga; exendin-4; glucagon-like peptide-1 receptor targeting; insulinoma.

Publication types

  • Randomized Controlled Trial
  • Research Support, Non-U.S. Gov't

MeSH terms

  • Adult
  • Cross-Over Studies
  • Diagnostic Imaging
  • Exenatide
  • Female
  • Gallium Radioisotopes / chemistry*
  • Glucose / chemistry
  • Heterocyclic Compounds, 1-Ring / chemistry*
  • Humans
  • Immunohistochemistry
  • Insulinoma / diagnostic imaging*
  • Male
  • Middle Aged
  • Multimodal Imaging
  • Peptides / chemistry*
  • Pilot Projects
  • Positron-Emission Tomography*
  • Tomography, Emission-Computed, Single-Photon
  • Tomography, X-Ray Computed*
  • Venoms / chemistry*
  • Whole Body Imaging

Substances

  • Gallium Radioisotopes
  • Heterocyclic Compounds, 1-Ring
  • Peptides
  • Venoms
  • 1,4,7,10-tetraazacyclododecane- 1,4,7,10-tetraacetic acid
  • Exenatide
  • Glucose