Cyclin-dependent kinase 2 (CDK2) is a key mediator for EGF-induced cell transformation mediated through the ELK4/c-Fos signaling pathway

Oncogene. 2016 Mar 3;35(9):1170-9. doi: 10.1038/onc.2015.175. Epub 2015 Jun 1.

Abstract

Cyclin-dependent kinase 2 (CDK2) is a known regulator in the cell cycle control of the G1/S and S/G2 transitions. However, the role of CDK2 in tumorigenesis is controversial. Evidence from knockout mice as well as colon cancer cell lines indicated that CDK2 is dispensable for cell proliferation. In this study, we found that ectopic CDK2 enhances Ras (G12V)-induced foci formation and knocking down CDK2 expression markedly decreases epidermal growth factor (EGF)-induced cell transformation mediated through the downregulation of c-fos expression. Interestingly, CDK2 directly phosphorylates ELK4 at Thr194 and Ser387 and regulates the ELK4 transcriptional activity, which serves as a mechanism to regulate c-fos expression. In addition, ELK4 is overexpressed in melanoma and knocking down the ELK4 or CDK2 expression significantly attenuated the malignant phenotype of melanoma cells. Taken together, our study reveals a novel function of CDK2 in EGF-induced cell transformation and the associated signal transduction pathways. This indicates that CDK2 is a useful molecular target for the chemoprevention and therapy against skin cancer.

Publication types

  • Research Support, N.I.H., Extramural
  • Research Support, Non-U.S. Gov't

MeSH terms

  • Animals
  • Cell Cycle / genetics
  • Cell Line
  • Cell Proliferation
  • Cell Transformation, Neoplastic / genetics
  • Cyclin-Dependent Kinase 2 / biosynthesis
  • Cyclin-Dependent Kinase 2 / genetics*
  • Epidermal Growth Factor / genetics
  • Epidermal Growth Factor / metabolism
  • Humans
  • Melanoma / genetics*
  • Melanoma / pathology
  • Mice
  • Phosphorylation
  • Proto-Oncogene Proteins c-fos / biosynthesis*
  • Transcriptional Activation / genetics
  • ets-Domain Protein Elk-4 / biosynthesis*
  • ets-Domain Protein Elk-4 / genetics

Substances

  • ELK4 protein, human
  • Proto-Oncogene Proteins c-fos
  • ets-Domain Protein Elk-4
  • Epidermal Growth Factor
  • CDK2 protein, human
  • Cyclin-Dependent Kinase 2