Precision-guided antimicrobial peptide as a targeted modulator of human microbial ecology

Proc Natl Acad Sci U S A. 2015 Jun 16;112(24):7569-74. doi: 10.1073/pnas.1506207112. Epub 2015 Jun 1.

Abstract

One major challenge to studying human microbiome and its associated diseases is the lack of effective tools to achieve targeted modulation of individual species and study its ecological function within multispecies communities. Here, we show that C16G2, a specifically targeted antimicrobial peptide, was able to selectively kill cariogenic pathogen Streptococcus mutans with high efficacy within a human saliva-derived in vitro oral multispecies community. Importantly, a significant shift in the overall microbial structure of the C16G2-treated community was revealed after a 24-h recovery period: several bacterial species with metabolic dependency or physical interactions with S. mutans suffered drastic reduction in their abundance, whereas S. mutans' natural competitors, including health-associated Streptococci, became dominant. This study demonstrates the use of targeted antimicrobials to modulate the microbiome structure allowing insights into the key community role of specific bacterial species and also indicates the therapeutic potential of C16G2 to achieve a healthy oral microbiome.

Keywords: dental caries; human microbiome; oral microbiota; targeted antimicrobial.

Publication types

  • Research Support, N.I.H., Extramural
  • Research Support, Non-U.S. Gov't

MeSH terms

  • Adult
  • Anti-Bacterial Agents / pharmacology
  • Antimicrobial Cationic Peptides / pharmacology*
  • Biofilms / drug effects
  • Biofilms / growth & development
  • Dental Caries / microbiology
  • Humans
  • Microbial Sensitivity Tests
  • Microbiota / drug effects*
  • Mouth / microbiology
  • Saliva / microbiology
  • Streptococcus mutans / drug effects*
  • Streptococcus mutans / pathogenicity
  • Streptococcus mutans / physiology*

Substances

  • Anti-Bacterial Agents
  • Antimicrobial Cationic Peptides