On-the-Road Driving Performance the Morning after Bedtime Use of Suvorexant 20 and 40 mg: A Study in Non-Elderly Healthy Volunteers

Sleep. 2015 Nov 1;38(11):1803-13. doi: 10.5665/sleep.5168.

Abstract

Study objective: To evaluate next-morning driving performance in adults younger than 65 years, after single and repeated doses of suvorexant 20 and 40 mg.

Design: Double-blind, placebo-controlled, 4-period crossover study.

Setting: Maastricht University, The Netherlands.

Participants: 28 healthy volunteers (15 females), aged 23 to 64 years.

Interventions: Suvorexant (20 and 40 mg) for 8 consecutive nights; zopiclone 7.5 mg nightly on day 1 and 8; placebo.

Measurements: Performance on day 2 and 9 (9 h after dosing) using a one-hour standardized highway driving test in normal traffic, measuring standard deviation of lateral position (SDLP). Drug-placebo changes in SDLP > 2.4 cm were considered to reflect meaningful driving impairment.

Results: Mean drug-placebo changes in SDLP following suvorexant 20 and 40 mg were 1.01 and 1.66 cm on day 2, and 0.48 and 1.31 cm on Day 9, respectively. The 90% CIs of these changes were all below 2.4 cm. Symmetry analysis showed that more subjects had SDLP changes > 2.4 cm than < -2.4 cm following suvorexant 20 and 40 mg on day 2, and following suvorexant 40 mg on day 9. Four female subjects requested that a total of 5 driving tests--all following suvorexant--stop prematurely due to self-reported somnolence.

Conclusions: As assessed by mean changes in standard deviation of lateral position (SDLP), there was no clinically meaningful residual effect of suvorexant in doses of 20 and 40 mg on next-morning driving (9 h after bedtime dosing) in healthy subjects < 65 years old. There may be some individuals who experience next-day effects, as suggested by individual changes in SDLP and prematurely stopped tests.

Clinical trial registration: clinicaltrials.gov NCT01311882.

Keywords: DSST; balance; driving; hypnotics; memory; orexin antagonist; plasma concentrations; suvorexant; zopiclone.

Publication types

  • Randomized Controlled Trial
  • Research Support, Non-U.S. Gov't

MeSH terms

  • Adult
  • Automobile Driving / psychology*
  • Azabicyclo Compounds / administration & dosage
  • Azabicyclo Compounds / pharmacology
  • Azepines / administration & dosage*
  • Azepines / pharmacology*
  • Cross-Over Studies
  • Double-Blind Method
  • Female
  • Healthy Volunteers*
  • Humans
  • Individuality
  • Male
  • Middle Aged
  • Netherlands
  • Piperazines / administration & dosage
  • Piperazines / pharmacology
  • Psychomotor Performance / drug effects
  • Self Report
  • Sleep Aids, Pharmaceutical / administration & dosage*
  • Sleep Aids, Pharmaceutical / pharmacology*
  • Sleep Stages / drug effects
  • Sleep Stages / physiology
  • Triazoles / administration & dosage*
  • Triazoles / pharmacology*
  • Young Adult

Substances

  • Azabicyclo Compounds
  • Azepines
  • Piperazines
  • Sleep Aids, Pharmaceutical
  • Triazoles
  • zopiclone
  • suvorexant

Associated data

  • ClinicalTrials.gov/NCT01311882