The toxic effects of Bisphenol A on the mouse spermatocyte GC-2 cell line: the role of the Ca2+-calmodulin-Ca2+/calmodulin-dependent protein kinase II axis

J Appl Toxicol. 2015 Nov;35(11):1271-7. doi: 10.1002/jat.3188. Epub 2015 Jun 18.

Abstract

Bisphenol A (BPA), an endocrine-disrupting chemical (EDC), is known to induce male reproductive toxicity in rodents. However, its toxic effects on the germ cells are still poorly understood. It has been proposed that Ca(2+) homeostasis and Ca(2+) sensors, including calmodulin (CaM) and calmodulin-dependent protein kinase II (CaMKII), play critical roles in spermatogenesis. Therefore, in the present study, we aimed to investigate whether a perturbation in Ca(2+)-CaM-CaMKII signaling was involved in the BPA-induced injury to mouse spermatocyte GC-2spd (ts) (GC-2) cells. Our results showed that BPA (range from 0.2 to 20 μM) induced obvious GC-2 cell injury, including decreased cell viability, the release of mitochondrial cytochrome c and the activation of caspase-3. However, these processes could be partially abrogated by pretreatment with a Ca(2+) chelator (BAPTA/AM), a CaM antagonist (W7) or a CaMKII inhibitor (KN93). These results, taken together, indicate that BPA exposure contributes to male germ cell injury, which may be partially mediated through a perturbation in Ca(2+)/CaM/CaMKII signaling and the mitochondrial apoptotic process.

Keywords: Bisphenol A; GC-2 cells; apoptosis; calcium; calcium/calmodulin-dependent protein kinase II; calmodulin.

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • Animals
  • Apoptosis / drug effects
  • Benzhydryl Compounds / toxicity*
  • Calcium-Calmodulin-Dependent Protein Kinase Type 2 / genetics
  • Calcium-Calmodulin-Dependent Protein Kinase Type 2 / metabolism*
  • Calmodulin / genetics
  • Calmodulin / metabolism*
  • Caspase 3 / genetics
  • Caspase 3 / metabolism
  • Cell Line
  • Cell Survival / drug effects
  • Cytochromes c / genetics
  • Cytochromes c / metabolism
  • Endocrine Disruptors / toxicity
  • Male
  • Mice
  • Mitochondria / drug effects
  • Phenols / toxicity*
  • Signal Transduction
  • Spermatocytes / cytology
  • Spermatocytes / drug effects*

Substances

  • Benzhydryl Compounds
  • Calmodulin
  • Endocrine Disruptors
  • Phenols
  • Cytochromes c
  • Calcium-Calmodulin-Dependent Protein Kinase Type 2
  • Casp3 protein, mouse
  • Caspase 3
  • bisphenol A