Efficiency and safety of subconjunctival injection of anti-VEGF agent - bevacizumab - in treating dry eye

Drug Des Devel Ther. 2015 Jun 12:9:3043-50. doi: 10.2147/DDDT.S85529. eCollection 2015.

Abstract

Purpose: Dry eye is a chronic inflammatory ocular surface disease with high prevalence. The current therapies for dry eye remain to be unspecific and notcomprehensive. This study aims to explore safety and efficacy of a novel treatment - subconjunctival injection of bevacizumab - in dry eye patients.

Methods: Sixty-four eyes of 32 dry eye patients received subconjunctival injection of 100 μL 25 mg/mL bevacizumab. Dry eye symptoms, signs (corrected visual acuity, intraocular pressure, conjunctival vascularity, corneal staining, tear break-up time, Marx line score, and blood pressure), and conjunctival impression cytology were evaluated 3 days before and 1 week, 1 month, and 3 months after injection.

Results: Significant improvements were observed in dry eye symptoms, tear break-up time, and conjunctival vascularization area at all the visits after injection compared to the baseline (P<0.05). The density of the goblet cell increased significantly at 1 month and 3 months after injection (P<0.05). There was no visual and systemic threat observed in any patient.

Conclusion: Subconjunctival injection of 100 μL 25 mg/mL bevacizumab is a safe and efficient treatment for ocular surface inflammation of dry eye disease.

Keywords: anti-VEGF; bevacizumab; dry eye; ocular surface inflammation; subconjunctival.

Publication types

  • Clinical Trial

MeSH terms

  • Adolescent
  • Adult
  • Aged
  • Aged, 80 and over
  • Angiogenesis Inhibitors / administration & dosage*
  • Angiogenesis Inhibitors / adverse effects
  • Angiogenesis Inhibitors / therapeutic use*
  • Bevacizumab / administration & dosage*
  • Bevacizumab / adverse effects
  • Bevacizumab / therapeutic use*
  • Conjunctiva / blood supply
  • Conjunctiva / pathology
  • Cornea / pathology
  • Dry Eye Syndromes / drug therapy*
  • Female
  • Goblet Cells / drug effects
  • Humans
  • Injections
  • Male
  • Meibomian Glands / pathology
  • Middle Aged
  • Regional Blood Flow / drug effects
  • Tears / drug effects
  • Treatment Outcome
  • Vascular Endothelial Growth Factor A / antagonists & inhibitors*
  • Young Adult

Substances

  • Angiogenesis Inhibitors
  • Vascular Endothelial Growth Factor A
  • Bevacizumab