Enhancement of the thermostability of Streptomyces kathirae SC-1 tyrosinase by rational design and empirical mutation

Enzyme Microb Technol. 2015 Sep:77:54-60. doi: 10.1016/j.enzmictec.2015.06.002. Epub 2015 Jun 11.

Abstract

This study aimed to improve the thermostability of a newly cloned tyrosinase from Streptomyces kathirae SC-1. The POPMuSiC algorithm was applied to predict the folding free energy change (ΔDG) of amino acid substitution. Site-directed mutagenesis was used to construct mutants (Q7K, G234P, and Q7K/G234P), and the mutant, and wild-type enzymes were expressed in Escherichia coli (DE3). Compared to the wild-type tyrosinase, all three mutant enzymes showed improved thermal properties. The mutant with combined substitution (Q7K/G234P) showed the most pronounced shifts in temperature optima, about 10 °C upward, and the half-life for thermal inactivation at 60 °C, and melting temperatures were increased by 3 times and approximately 10 °C, respectively. Finally, the mechanisms responsible for the increased thermostability were analyzed through comparative analysis of structure models. The structure-based rational design strategies in this study may also provide further insight into the thermostability of other industrial enzymes and suggest further potential industrial applications.

Keywords: POPMuSiC; Site-directed mutagenesis; Thermostability; Tyrosinase.

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • Amino Acid Substitution
  • Bacterial Proteins / chemistry
  • Bacterial Proteins / genetics*
  • Bacterial Proteins / metabolism*
  • Catalytic Domain / genetics
  • Enzyme Stability / genetics
  • Hydrogen-Ion Concentration
  • Kinetics
  • Models, Molecular
  • Monophenol Monooxygenase / chemistry
  • Monophenol Monooxygenase / genetics*
  • Monophenol Monooxygenase / metabolism*
  • Mutagenesis, Site-Directed
  • Mutant Proteins / chemistry
  • Mutant Proteins / genetics
  • Mutant Proteins / metabolism
  • Protein Conformation
  • Recombinant Proteins / chemistry
  • Recombinant Proteins / genetics
  • Recombinant Proteins / metabolism
  • Streptomyces / enzymology*
  • Streptomyces / genetics*
  • Temperature

Substances

  • Bacterial Proteins
  • Mutant Proteins
  • Recombinant Proteins
  • Monophenol Monooxygenase